TRANSPORT CHARACTERISTICS OF CEFTIBUTEN, A NEW ORAL CEPHEM, IN RAT INTESTINAL BRUSH-BORDER MEMBRANE-VESICLES - RELATIONSHIP TO OLIGOPEPTIDE AND AMINO BETA-LACTAM TRANSPORT

被引:61
作者
MURANUSHI, N [1 ]
YOSHIKAWA, T [1 ]
YOSHIDA, M [1 ]
OGUMA, T [1 ]
HIRANO, K [1 ]
YAMADA, H [1 ]
机构
[1] SHIONOGI & CO LTD,SHIONOGI RES LAB,FUKUSHIMA KU,OSAKA 553,JAPAN
关键词
D O I
10.1023/A:1015946407709
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
收藏
页码:308 / 312
页数:5
相关论文
共 21 条
[1]   SODIUM ION-COUPLED UPTAKE OF TAUROCHOLATE BY INTESTINAL BRUSH-BORDER MEMBRANE-VESICLES [J].
BEESLEY, RC ;
FAUST, RG .
BIOCHEMICAL JOURNAL, 1979, 178 (02) :299-303
[2]  
CRANE RK, 1962, FED PROC, V21, P891
[3]  
GANAPATHY V, 1983, J BIOL CHEM, V258, P4189
[4]  
HIRANO K, 1986, 26TH INT C ANT AG CH
[5]   UPTAKE OF AMINO BETA-LACTAM ANTIBIOTICS INTO RAT INTESTINAL BRUSH-BORDER MEMBRANE-VESICLES [J].
ISEKI, K ;
IEMURA, A ;
MIYAZAKI, K ;
ARITA, T .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1985, 37 (05) :374-375
[6]   MODIFIED PROCEDURE FOR RAPID PREPARATION OF EFFICIENTLY TRANSPORTING VESICLES FROM SMALL INTESTINAL BRUSH-BORDER MEMBRANES - THEIR USE IN INVESTIGATING SOME PROPERTIES OF D-GLUCOSE AND CHOLINE TRANSPORT-SYSTEMS [J].
KESSLER, M ;
ACUTO, O ;
STORELLI, C ;
MURER, H ;
MULLER, M ;
SEMENZA, G .
BIOCHIMICA ET BIOPHYSICA ACTA, 1978, 506 (01) :136-154
[7]  
KIMURA T, 1983, J PHARMACOBIO-DYNAM, V6, P246
[8]   TRANSPORT OF CEFADROXIL, AN AMINOCEPHALOSPORIN ANTIBIOTIC, ACROSS THE SMALL INTESTINAL BRUSH-BORDER MEMBRANE [J].
KIMURA, T ;
YAMAMOTO, T ;
ISHIZUKA, R ;
SEZAKI, H .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (01) :81-84
[9]  
KIMURA T, 1978, Journal of Pharmacobio-Dynamics, V1, P262
[10]   DIRECT MEASUREMENT BY PH-MICROELECTRODE OF PH MICROCLIMATE IN RAT PROXIMAL JEJUNUM [J].
LUCAS, ML ;
SCHNEIDER, W ;
HABERICH, FJ ;
BLAIR, JA .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1975, 192 (1106) :39-48