SYNTHESIS AND BIOLOGICAL EVALUATION OF 14-ALKOXYMORPHINANS .2. (-)-N-(CYCLOPROPYLMETHYL)-4,14-DIMETHOXYMORPHINAN-6-ONE, A SELECTIVE MU-OPIOID RECEPTOR ANTAGONIST

被引:93
作者
SCHMIDHAMMER, H
BURKARD, WP
EGGSTEINAEPPLI, L
SMITH, CFC
机构
[1] F HOFFMANN LA ROCHE & CO LTD, PHARMACEUT RES DEPT, CH-4002 BASEL, SWITZERLAND
[2] RECKITT & COLMAN LTD, DIV PHARMACEUT, HULL HU8 7DS, N HUMBERSIDE, ENGLAND
关键词
D O I
10.1021/jm00122a021
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:418 / 421
页数:4
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