INHIBITION OF MONO-OXYGENASE AND OXIDASE ACTIVITY OF RAT-HEPATIC CYTOCHROME-P-450 BY H2-RECEPTOR BLOCKERS

被引:51
作者
BAST, A
SAVENIJECHAPEL, EM
KROES, BH
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关键词
D O I
10.3109/00498258409151428
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:399 / 408
页数:10
相关论文
共 23 条
[1]  
BAST A, 1983, RES COMMUN CHEM PATH, V40, P391
[2]   SPECTRAL INTERACTION OF ORPHENADRINE AND ITS METABOLITES WITH OXIDIZED AND REDUCED HEPATIC-MICROSOMAL CYTOCHROME-P-450 IN THE RAT [J].
BAST, A ;
NOORDHOEK, J .
BIOCHEMICAL PHARMACOLOGY, 1982, 31 (17) :2745-2753
[3]   CYTOCHROME-P450 OXIDASE ACTIVITY AND ITS ROLE IN NADPH DEPENDENT LIPID-PEROXIDATION [J].
BAST, A ;
BRENNINKMEIJER, JW ;
SAVENIJECHAPEL, EM ;
NOORDHOEK, J .
FEBS LETTERS, 1983, 151 (02) :185-188
[4]   CALCULATION OF COMPETITIVE-INHIBITION OF SUBSTRATE BINDING TO CYTOCHROME-P-450 ILLUSTRATED BY THE INTERACTION OF D,L-PROPRANOLOL WITH D,L-HEXOBARBITAL [J].
BAST, A ;
NOORDHOEK, J .
BIOCHEMICAL PHARMACOLOGY, 1980, 29 (05) :747-751
[5]   FURTHER-STUDIES ON THE DISSOCIATION OF THE ISOSAFROLE METABOLITE-CYTOCHROME-P-450 COMPLEX [J].
DICKINS, M ;
ELCOMBE, CR ;
MOLONEY, SJ ;
NETTER, KJ ;
BRIDGES, JW .
BIOCHEMICAL PHARMACOLOGY, 1979, 28 (02) :231-238
[6]  
DREW R, 1981, RES COMMUN CHEM PATH, V33, P81
[7]  
Estabrook RW., 1972, METHODS PHARM, Vvol 2, P303
[8]   INTERACTION OF ISOSAFROLE INVIVO WITH RAT HEPATIC MICROSOMAL CYTOCHROME-P-450 FOLLOWING TREATMENT WITH PHENOBARBITONE OR 20-METHYLCHOLANTHRENE [J].
FENNELL, TR ;
DICKINS, M ;
BRIDGES, JW .
BIOCHEMICAL PHARMACOLOGY, 1979, 28 (08) :1427-1429
[9]   HEXOBARBITAL-BINDING, HYDROXYLATION AND HEXOBARBITAL-DEPENDENT HYDROGEN-PEROXIDE PRODUCTION IN HEPATIC MICROSOMES OF GUINEA-PIG, RAT AND RABBIT [J].
HEINEMEYER, G ;
NIGAM, S ;
HILDEBRANDT, AG .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 314 (02) :201-210
[10]  
Hildebrandt A G, 1978, Methods Enzymol, V52, P342