EFFECTS OF BETA-ADRENOCEPTOR ANTAGONIST ADMINISTRATION ON BETA-2-ADRENOCEPTOR DENSITY IN HUMAN-LYMPHOCYTES - THE ROLE OF THE INTRINSIC SYMPATHOMIMETIC ACTIVITY

被引:50
作者
BRODDE, OE [1 ]
DAUL, A [1 ]
STUKA, N [1 ]
OHARA, N [1 ]
BORCHARD, U [1 ]
机构
[1] UNIV DUSSELDORF,INST PHARMACOL,D-4000 DUSSELDORF,FED REP GER
关键词
D O I
10.1007/BF00692910
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:417 / 422
页数:6
相关论文
共 17 条
[1]   ELEVATION OF BETA-ADRENERGIC-RECEPTOR DENSITY IN HUMAN-LYMPHOCYTES AFTER PROPRANOLOL ADMINISTRATION [J].
AARONS, RD ;
NIES, AS ;
GAL, J ;
HEGSTRAND, LR ;
MOLINOFF, PB .
JOURNAL OF CLINICAL INVESTIGATION, 1980, 65 (05) :949-957
[2]  
AARONS RD, 1982, J PHARMACOL EXP THER, V221, P439
[3]  
BOYUM A, 1968, SCAND J CLIN LAB INV, VS 21, P77
[4]   NO EVIDENCE FOR TEMPERATURE-DEPENDENT CHANGES IN THE PHARMACOLOGICAL SPECIFICITY OF BETA-1-ADRENOCEPTORS AND BETA-2-ADRENOCEPTORS IN RABBIT LUNG MEMBRANES [J].
BRODDE, OE ;
KUHLHOFF, F ;
ARROYO, J ;
PRYWARRA, A .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1983, 322 (01) :20-28
[5]   THE BETA-ADRENERGIC-RECEPTOR IN HUMAN-LYMPHOCYTES - SUBCLASSIFICATION BY THE USE OF A NEW RADIO-LIGAND, (+/-)-IODOCYANOPINDOLOL-125 [J].
BRODDE, OE ;
ENGEL, G ;
HOYER, D ;
BOCK, KD ;
WEBER, F .
LIFE SCIENCES, 1981, 29 (21) :2189-2198
[6]   COEXISTENCE OF BETA-1-ADRENOCEPTORS AND BETA-2-ADRENOCEPTORS IN HUMAN RIGHT ATRIUM - DIRECT IDENTIFICATION BY (+/-)-[I-125]IODOCYANOPINDOLOL BINDING [J].
BRODDE, OE ;
KARAD, K ;
ZERKOWSKI, HR ;
ROHM, N ;
REIDEMEISTER, JC .
CIRCULATION RESEARCH, 1983, 53 (06) :752-758
[7]  
DAUL A, 1984, NAUNYNSCHMIEDEBERG S, V325, pR264
[8]   COMPARISON OF CHANGES IN THE CHARACTERISTICS OF BETA-ADRENOCEPTORS AND RESPONSIVENESS OF HUMAN CIRCULATING LYMPHOCYTES DURING AND AFTER CHRONIC ADMINISTRATION OF PINDOLOL AND PROPRANOLOL [J].
GIUDICELLI, Y ;
LACASA, D ;
AGLI, B ;
LENEVEU, A .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1984, 26 (01) :7-12
[9]   RADIOLIGAND BINDING-STUDIES OF ADRENERGIC-RECEPTORS - NEW INSIGHTS INTO MOLECULAR AND PHYSIOLOGICAL REGULATION [J].
HOFFMAN, BB ;
LEFKOWITZ, RJ .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1980, 20 :581-608
[10]   EFFECTS OF DRUGS ON BETA-ADRENERGIC RECEPTORS ON HUMAN-LYMPHOCYTES [J].
MOLINOFF, PB ;
AARONS, RD .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1983, 5 :S63-S67