L-649,923,SODIUM (BETA-S-STAR,GAMMA-R-STAR)-4-(3-(4-ACETYL-3-HYDROXY-2-PROPYLPHENOXY)PROPYLTHIO)-GAMMA-HYDROXY-BETA-METHYLBENZENEBUTANOATE, A SELECTIVE, ORALLY ACTIVE LEUKOTRIENE RECEPTOR ANTAGONIST

被引：76

作者：

JONES, TR ^{[1
]}

YOUNG, R ^{[1
]}

CHAMPION, E ^{[1
]}

CHARETTE, L ^{[1
]}

DENIS, D ^{[1
]}

FORDHUTCHINSON, AW ^{[1
]}

FRENETTE, R ^{[1
]}

GAUTHIER, JY ^{[1
]}

GUINDON, Y ^{[1
]}

KAKUSHIMA, M ^{[1
]}

MASSON, P ^{[1
]}

MCFARLANE, C ^{[1
]}

PIECHUTA, H ^{[1
]}

ROKACH, J ^{[1
]}

ZAMBONI, R ^{[1
]}

DEHAVEN, RN ^{[1
]}

MAYCOCK, A ^{[1
]}

PONG, SS ^{[1
]}

机构：

[1] MERCK SHARP & DOHME RES LABS,DEPT BIOCHEM INFLAMMAT,RAHWAY,NJ 07065

来源：

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY | 1986年 / 64卷 / 08期

关键词：

D O I：

10.1139/y86-183

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：1068 / 1075

页数：8

共 44 条

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[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (06): : 3887 - 3891
[9] COMPARATIVE AIRWAY AND VASCULAR ACTIVITIES OF LEUKOTRIENE-C-1 AND LEUKOTRIENE-D INVIVO AND INVITRO
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[J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (07): : 4354 - 4358
[10] EVIDENCE FOR MULTIPLE LEUKOTRIENE-D4 RECEPTORS IN SMOOTH-MUSCLE
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[J]. LIFE SCIENCES, 1982, 31 (06) : 577 - 581

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