PALLADIUM IN CEPHALOSPORIN CHEMISTRY - AN INEXPENSIVE TRIFLATE REPLACEMENT FOR PALLADIUM ACETATE MEDIATED COUPLING REACTIONS

被引：35

作者：

ROTH, GP

SAPINO, C

机构：

[1] Bristol-Myers Squibb Company Pharmaceutical Research Institute, Wallingford, CT 06492

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 33期

关键词：

D O I：

10.1016/S0040-4039(00)79866-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

3-Fluorosulfonyloxy-3-cephems are easily prepared and subsequent palladium(0) catalyzed coupling with various vinylstannanes proceeds in excellent yields with stereospecific transfer of the alkene fragment.

引用

页码：4073 / 4076

页数：4

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