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ACTIVITY OF AROMATIC SUBSTITUTED PHENYLPIPERAZINES LACKING AFFINITY FOR DOPAMINE BINDING-SITES IN A PRECLINICAL TEST OF ANTIPSYCHOTIC EFFICACY
被引:74
作者
:
MARTIN, GE
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
MARTIN, GE
ELGIN, RJ
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
ELGIN, RJ
MATHIASEN, JR
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
MATHIASEN, JR
DAVIS, CB
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
DAVIS, CB
KESSLICK, JM
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
KESSLICK, JM
BALDY, WJ
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
BALDY, WJ
SHANK, RP
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
SHANK, RP
DISTEFANO, DL
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
DISTEFANO, DL
FEDDE, CL
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
FEDDE, CL
SCOTT, MK
论文数:
0
引用数:
0
h-index:
0
机构:
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
SCOTT, MK
机构
:
[1]
MCNEIL PHARMACEUT,DEPT BIOL RES,SPRING HOUSE,PA 19477
[2]
MCNEIL PHARMACEUT,DEPT MED CHEM,SPRING HOUSE,PA 19477
[3]
JANSSEN RES FDN WORLDWIDE,SPRING HOUSE,PA 19477
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1989年
/ 32卷
/ 05期
关键词
:
D O I
:
10.1021/jm00125a020
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:1052 / 1056
页数:5
相关论文
共 28 条
[1]
ASH ASF, 1964, Patent No. 3133056
[2]
BYSOUTH PT, 1969, Patent No. 6804082
[3]
SEROTONIN FUNCTION IN ANXIETY .2. EFFECTS OF THE SEROTONIN AGONIST MCPP IN PANIC DISORDER PATIENTS AND HEALTHY-SUBJECTS
CHARNEY, DS
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
CHARNEY, DS
WOODS, SW
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
WOODS, SW
GOODMAN, WK
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引用数:
0
h-index:
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YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
GOODMAN, WK
HENINGER, GR
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
HENINGER, GR
[J].
PSYCHOPHARMACOLOGY,
1987,
92
(01)
: 14
-
24
[4]
CENTRAL SEROTONIN-LIKE ACTIVITY OF "6-CHLORO-2-[1-PIPERAZINYL]-PYRAZINE (CPP-MK-212)
CLINESCHMIDT, BV
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,W POINT,PA 19486
MERCK INST THERAPEUT RES,W POINT,PA 19486
CLINESCHMIDT, BV
MCGUFFIN, JC
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,W POINT,PA 19486
MERCK INST THERAPEUT RES,W POINT,PA 19486
MCGUFFIN, JC
PFLUEGER, AB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,W POINT,PA 19486
MERCK INST THERAPEUT RES,W POINT,PA 19486
PFLUEGER, AB
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1977,
44
(01)
: 65
-
74
[5]
INVITRO RECEPTOR SPECIFICITY OF THE 5HT-1A SELECTIVE PHENYLPIPERAZINE, LY165163
COHEN, ML
论文数:
0
引用数:
0
h-index:
0
COHEN, ML
MASON, N
论文数:
0
引用数:
0
h-index:
0
MASON, N
SCHENCK, KW
论文数:
0
引用数:
0
h-index:
0
SCHENCK, KW
[J].
LIFE SCIENCES,
1986,
39
(25)
: 2441
-
2446
[6]
DIFFERENTIAL EFFECTS OF NEUROLEPTIC AND OTHER PSYCHOTROPIC AGENTS ON ACQUISITION OF AVOIDANCE IN RATS
DAVIDSON, AB
论文数:
0
引用数:
0
h-index:
0
机构:
SMITH KLINE & FRENCH LABS,DEPT PHARMACOL,PHILADELPHIA,PA
SMITH KLINE & FRENCH LABS,DEPT PHARMACOL,PHILADELPHIA,PA
DAVIDSON, AB
WEIDLEY, E
论文数:
0
引用数:
0
h-index:
0
机构:
SMITH KLINE & FRENCH LABS,DEPT PHARMACOL,PHILADELPHIA,PA
SMITH KLINE & FRENCH LABS,DEPT PHARMACOL,PHILADELPHIA,PA
WEIDLEY, E
[J].
LIFE SCIENCES,
1976,
18
(11)
: 1279
-
1284
[7]
STRUCTURAL RELATIONSHIPS IN THE INHIBITION OF [SEROTONIN-H-3 BINDING TO RAT-BRAIN MEMBRANES INVITRO BY 1-PHENYL-PIPERAZINES
FULLER, RW
论文数:
0
引用数:
0
h-index:
0
FULLER, RW
MASON, NR
论文数:
0
引用数:
0
h-index:
0
MASON, NR
MOLLOY, BB
论文数:
0
引用数:
0
h-index:
0
MOLLOY, BB
[J].
BIOCHEMICAL PHARMACOLOGY,
1980,
29
(05)
: 833
-
835
[8]
EFFECT OF 1-(M-TRIFLUOROMETHYLPHENYL)-PIPERAZINE ON SEROTONIN-H-3 BINDING TO MEMBRANES FROM RAT-BRAIN INVITRO AND ON SEROTONIN TURNOVER IN RAT-BRAIN INVIVO
FULLER, RW
论文数:
0
引用数:
0
h-index:
0
FULLER, RW
SNODDY, HD
论文数:
0
引用数:
0
h-index:
0
SNODDY, HD
MASON, NR
论文数:
0
引用数:
0
h-index:
0
MASON, NR
MOLLOY, BB
论文数:
0
引用数:
0
h-index:
0
MOLLOY, BB
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1978,
52
(01)
: 11
-
16
[9]
CENTRAL SEROTONIN RECEPTORS AS TARGETS FOR DRUG RESEARCH
GLENNON, RA
论文数:
0
引用数:
0
h-index:
0
GLENNON, RA
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1987,
30
(01)
: 1
-
12
[10]
BIOACTIVE CONFORMATION OF 1-ARYLPIPERAZINES AT CENTRAL SEROTONIN RECEPTORS
HUFF, JR
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
HUFF, JR
KING, SW
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
KING, SW
SAARI, WS
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
SAARI, WS
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
SPRINGER, JP
MARTIN, GE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
MARTIN, GE
WILLIAMS, M
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
WILLIAMS, M
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1985,
28
(07)
: 945
-
948
←
1
2
3
→
共 28 条
[1]
ASH ASF, 1964, Patent No. 3133056
[2]
BYSOUTH PT, 1969, Patent No. 6804082
[3]
SEROTONIN FUNCTION IN ANXIETY .2. EFFECTS OF THE SEROTONIN AGONIST MCPP IN PANIC DISORDER PATIENTS AND HEALTHY-SUBJECTS
CHARNEY, DS
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
CHARNEY, DS
WOODS, SW
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
WOODS, SW
GOODMAN, WK
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
GOODMAN, WK
HENINGER, GR
论文数:
0
引用数:
0
h-index:
0
机构:
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
YALE UNIV,SCH MED,DEPT PSYCHIAT,NEW HAVEN,CT 06510
HENINGER, GR
[J].
PSYCHOPHARMACOLOGY,
1987,
92
(01)
: 14
-
24
[4]
CENTRAL SEROTONIN-LIKE ACTIVITY OF "6-CHLORO-2-[1-PIPERAZINYL]-PYRAZINE (CPP-MK-212)
CLINESCHMIDT, BV
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,W POINT,PA 19486
MERCK INST THERAPEUT RES,W POINT,PA 19486
CLINESCHMIDT, BV
MCGUFFIN, JC
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,W POINT,PA 19486
MERCK INST THERAPEUT RES,W POINT,PA 19486
MCGUFFIN, JC
PFLUEGER, AB
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK INST THERAPEUT RES,W POINT,PA 19486
MERCK INST THERAPEUT RES,W POINT,PA 19486
PFLUEGER, AB
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1977,
44
(01)
: 65
-
74
[5]
INVITRO RECEPTOR SPECIFICITY OF THE 5HT-1A SELECTIVE PHENYLPIPERAZINE, LY165163
COHEN, ML
论文数:
0
引用数:
0
h-index:
0
COHEN, ML
MASON, N
论文数:
0
引用数:
0
h-index:
0
MASON, N
SCHENCK, KW
论文数:
0
引用数:
0
h-index:
0
SCHENCK, KW
[J].
LIFE SCIENCES,
1986,
39
(25)
: 2441
-
2446
[6]
DIFFERENTIAL EFFECTS OF NEUROLEPTIC AND OTHER PSYCHOTROPIC AGENTS ON ACQUISITION OF AVOIDANCE IN RATS
DAVIDSON, AB
论文数:
0
引用数:
0
h-index:
0
机构:
SMITH KLINE & FRENCH LABS,DEPT PHARMACOL,PHILADELPHIA,PA
SMITH KLINE & FRENCH LABS,DEPT PHARMACOL,PHILADELPHIA,PA
DAVIDSON, AB
WEIDLEY, E
论文数:
0
引用数:
0
h-index:
0
机构:
SMITH KLINE & FRENCH LABS,DEPT PHARMACOL,PHILADELPHIA,PA
SMITH KLINE & FRENCH LABS,DEPT PHARMACOL,PHILADELPHIA,PA
WEIDLEY, E
[J].
LIFE SCIENCES,
1976,
18
(11)
: 1279
-
1284
[7]
STRUCTURAL RELATIONSHIPS IN THE INHIBITION OF [SEROTONIN-H-3 BINDING TO RAT-BRAIN MEMBRANES INVITRO BY 1-PHENYL-PIPERAZINES
FULLER, RW
论文数:
0
引用数:
0
h-index:
0
FULLER, RW
MASON, NR
论文数:
0
引用数:
0
h-index:
0
MASON, NR
MOLLOY, BB
论文数:
0
引用数:
0
h-index:
0
MOLLOY, BB
[J].
BIOCHEMICAL PHARMACOLOGY,
1980,
29
(05)
: 833
-
835
[8]
EFFECT OF 1-(M-TRIFLUOROMETHYLPHENYL)-PIPERAZINE ON SEROTONIN-H-3 BINDING TO MEMBRANES FROM RAT-BRAIN INVITRO AND ON SEROTONIN TURNOVER IN RAT-BRAIN INVIVO
FULLER, RW
论文数:
0
引用数:
0
h-index:
0
FULLER, RW
SNODDY, HD
论文数:
0
引用数:
0
h-index:
0
SNODDY, HD
MASON, NR
论文数:
0
引用数:
0
h-index:
0
MASON, NR
MOLLOY, BB
论文数:
0
引用数:
0
h-index:
0
MOLLOY, BB
[J].
EUROPEAN JOURNAL OF PHARMACOLOGY,
1978,
52
(01)
: 11
-
16
[9]
CENTRAL SEROTONIN RECEPTORS AS TARGETS FOR DRUG RESEARCH
GLENNON, RA
论文数:
0
引用数:
0
h-index:
0
GLENNON, RA
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1987,
30
(01)
: 1
-
12
[10]
BIOACTIVE CONFORMATION OF 1-ARYLPIPERAZINES AT CENTRAL SEROTONIN RECEPTORS
HUFF, JR
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
HUFF, JR
KING, SW
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
KING, SW
SAARI, WS
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
SAARI, WS
SPRINGER, JP
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
SPRINGER, JP
MARTIN, GE
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
MARTIN, GE
WILLIAMS, M
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,MERCK INST THERAPEUT RES,W POINT,PA 19486
WILLIAMS, M
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1985,
28
(07)
: 945
-
948
←
1
2
3
→