TISSUE-RESPONSE SELECTIVITY OF CALCIUM-ANTAGONISTS IS NOT DUE TO HETEROGENEITY OF [NITRENDIPINE-H-3 BINDING-SITES

被引:51
作者
BRISTOW, MR
GINSBURG, R
LASER, JA
MCAULEY, BJ
MINOBE, W
机构
关键词
D O I
10.1111/j.1476-5381.1984.tb10765.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
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页码:309 / 320
页数:12
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共 40 条
[1]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[2]  
BELLEMANN P, 1981, ARZNEIMITTEL-FORSCH, V31-2, P2064
[3]  
BELLEMANN P, 1982, ARZNEIMITTEL-FORSCH, V32-1, P361
[4]   HIGH-AFFINITY BINDING OF A CALCIUM-CHANNEL ANTAGONIST TO SMOOTH AND CARDIAC-MUSCLE [J].
BOLGER, GT ;
GENGO, PJ ;
LUCHOWSKI, EM ;
SIEGEL, H ;
TRIGGLE, DJ ;
JANIS, RA .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 104 (04) :1604-1609
[5]  
BRISTOW MR, 1982, CIRCULATION, V66, P95
[6]   DECREASED CATECHOLAMINE SENSITIVITY AND BETA-ADRENERGIC-RECEPTOR DENSITY IN FAILING HUMAN HEARTS [J].
BRISTOW, MR ;
GINSBURG, R ;
MINOBE, W ;
CUBICCIOTTI, RS ;
SAGEMAN, WS ;
LURIE, K ;
BILLINGHAM, ME ;
HARRISON, DC ;
STINSON, EB .
NEW ENGLAND JOURNAL OF MEDICINE, 1982, 307 (04) :205-211
[7]   EFFECT OF DIAZOXIDE, VERAPAMIL AND COMPOUND D600 ON ISOPROTERENOL AND CALCIUM-MEDIATED DOSE-RESPONSE RELATIONSHIPS IN ISOLATED RABBIT ATRIUM [J].
BRISTOW, MR ;
GREEN, RD .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1977, 45 (03) :267-279
[8]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[9]   SIMULTANEOUS ANALYSIS OF FAMILIES OF SIGMOIDAL CURVES - APPLICATION TO BIOASSAY, RADIOLIGAND ASSAY, AND PHYSIOLOGICAL DOSE-RESPONSE CURVES [J].
DELEAN, A ;
MUNSON, PJ ;
RODBARD, D .
AMERICAN JOURNAL OF PHYSIOLOGY, 1978, 235 (02) :E97-E102
[10]   SPECIFIC BINDING OF [H-3]LABELED NITRENDIPINE TO MEMBRANES FROM CORONARY-ARTERIES AND HEART IN RELATION TO PHARMACOLOGICAL EFFECTS - PARADOXICAL STIMULATION BY DILTIAZEM [J].
DEPOVER, A ;
MATLIB, MA ;
LEE, SW ;
DUBE, GP ;
GRUPP, IL ;
GRUPP, G ;
SCHWARTZ, A .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1982, 108 (01) :110-117