THE SYNTHESIS OF 5-ARYLPYRROLO[3,2-B]PYRIDINES AND 7-ARYLPYRROLO[3,2-B]PYRIDINES - ADDITION OF 3-AMINOPYRROLES TO ARYL ENAMINONES

被引：8

作者：

BIRNBERG, GH

FANSHAWE, WJ

FRANCISCO, GD

EPSTEIN, JW

机构：

[1] Cardiovascular and Central Nervous System Disease Research Section, Medical Research Division, American Cyanamid Company, Lederle Laboratories, New York, 10965, Pearl River

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1995年 / 32卷 / 04期

关键词：

D O I：

10.1002/jhet.5570320433

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of 5-arylpyrrolo[3,2-b]pyridines 1 was synthesized by addition of 3-aminopyrroles to aryl enaminones. One example of a 7-arylpyrrolo[3,2-b]pyridine 2 was obtained as a minor product along with the 5-aryl isomer, by a modification of the reaction sequence.

引用

页码：1293 / 1298

页数：6

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