ASYMMETRIC-SYNTHESIS OF STEROIDAL TROGER BASE ANALOGS - X-RAY MOLECULAR-STRUCTURE OF METHYL 3-ALPHA,12-ALPHA-(6H,12H-5,11-METHANODIBENZO[B,F][1,5]DIAZOCINE-2,8-BISACETOXY)-5-BETA-CHOLAN-24-OATE

被引：29

作者：

MAITRA, U ^{[1
]}

BAG, BG ^{[1
]}

RAO, P ^{[1
]}

POWELL, D ^{[1
]}

机构：

[1] UNIV WISCONSIN,DEPT CHEM,MADISON,WI 53706

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1995年 / 16期

关键词：

D O I：

10.1039/p19950002049

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Cyclization of compound 5c in trifluoroacetic acid/hexamethylenetetramine produces Troger's base analogue 6c in 75% yield with 70% diastereoselectivity.

引用

页码：2049 / 2056

页数：8

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