THE INACTIVATION OF [MET5] ENKEPHALIN BY BESTATIN-SENSITIVE AMINOPEPTIDASE, CAPTOPRIL-SENSITIVE PEPTIDYL DIPEPTIDASE-A AND THIORPHAN-SENSITIVE ENDOPEPTIDASE-24.11 IN MOUSE VAS-DEFERENS

被引:30
作者
AOKI, K [1 ]
KAJIWARA, M [1 ]
OKA, T [1 ]
机构
[1] TOKAI UNIV,SCH MED,DEPT PHARMACOL,ISEHARA,KANAGAWA 25911,JAPAN
关键词
D O I
10.1254/jjp.40.297
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:297 / 302
页数:6
相关论文
共 12 条
[1]   THE ROLE OF BESTATIN-SENSITIVE AMINOPEPTIDASE, ANGIOTENSIN CONVERTING ENZYME AND THIORPHAN-SENSITIVE ENKEPHALINASE IN THE POTENCY OF ENKEPHALINS IN THE GUINEA-PIG ILEUM [J].
AOKI, K ;
KAJIWARA, M ;
OKA, T .
JAPANESE JOURNAL OF PHARMACOLOGY, 1984, 36 (01) :59-65
[2]  
EHRENPREIS S, 1978, CHARACTERISTICS FUNC, P417
[3]   ENKEPHALINASES [J].
GORENSTEIN, C ;
SNYDER, SH .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1980, 210 (1178) :123-132
[4]  
Hartsuck J. A., 1971, ENZYMES, V3, P1
[5]  
LEE CM, 1982, J BIOL CHEM, V257, P2043
[6]   HIGH-AFFINITY ENKEPHALIN-DEGRADING PEPTIDASE IN BRAIN IS INCREASED AFTER MORPHINE [J].
MALFROY, B ;
SWERTS, JP ;
GUYON, A ;
ROQUES, BP ;
SCHWARTZ, JC .
NATURE, 1978, 276 (5687) :523-526
[7]   SUBSTANCE-P AND [LEU]ENKEPHALIN ARE HYDROLYZED BY AN ENZYME IN PIG CAUDATE SYNAPTIC-MEMBRANES THAT IS IDENTICAL WITH THE ENDOPEPTIDASE OF KIDNEY MICROVILLI [J].
MATSAS, R ;
FULCHER, IS ;
KENNY, AJ ;
TURNER, AJ .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (10) :3111-3115
[8]   THE METABOLISM OF NEUROPEPTIDES - THE HYDROLYSIS OF PEPTIDES, INCLUDING ENKEPHALINS, TACHYKININS AND THEIR ANALOGS, BY ENDOPEPTIDASE-24-11 [J].
MATSAS, R ;
KENNY, AJ ;
TURNER, AJ .
BIOCHEMICAL JOURNAL, 1984, 223 (02) :433-440
[9]   STRUCTURE-ACTIVITY-RELATIONSHIPS OF ENKEPHALIN-LIKE PEPTIDES [J].
MORLEY, JS .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1980, 20 :81-110
[10]   EVIDENCE THAT DYNORPHIN-(1-13) ACTS AS AN AGONIST ON OPIOID K-RECEPTORS [J].
OKA, T ;
NEGISHI, K ;
SUDA, M ;
SAWA, A ;
FUJINO, M ;
WAKIMASU, M .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1982, 77 (2-3) :137-141