AMODIAQUINE AS A PRODRUG - IMPORTANCE OF METABOLITE(S) IN THE ANTIMALARIAL EFFECT OF AMODIAQUINE IN HUMANS

被引:102
作者
CHURCHILL, FC
PATCHEN, LC
CAMPBELL, CC
SCHWARTZ, IK
PHUC, ND
DICKINSON, CM
机构
关键词
D O I
10.1016/0024-3205(85)90285-1
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
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页码:53 / 62
页数:10
相关论文
共 11 条
[1]   DISPOSITION AND METABOLISM OF AMODIAQUINE IN SMALL MAMMALS [J].
BARROW, A .
XENOBIOTICA, 1974, 4 (11) :669-680
[2]  
BRODIE BB, 1947, J BIOL CHEM, V168, P319
[3]   EVALUATION OF AMODIAQUINE TREATMENT OF CHLOROQUINE-RESISTANT PLASMODIUM-FALCIPARUM MALARIA ON ZANZIBAR, 1982 [J].
CAMPBELL, CC ;
PAYNE, D ;
SCHWARTZ, IK ;
KHATIB, OJ .
AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, 1983, 32 (06) :1216-1220
[4]  
NGUYENDINH P, 1981, B WORLD HEALTH ORGAN, V59, P641
[5]   PLASMODIUM-FALCIPARUM INVITRO - DETERMINATION OF CHLOROQUINE SENSITIVITY OF 3 NEW STRAINS BY A MODIFIED 48-HOUR TEST [J].
NGUYENDINH, P ;
TRAGER, W .
AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, 1980, 29 (03) :339-342
[6]   TREATMENT OF PLASMODIUM-FALCIPARUM MALARIA WITH A COMBINATION OF AMODIAQUINE AND TETRACYCLINE IN CENTRAL THAILAND [J].
NOEYPATIMANOND, S ;
MALIKUL, S ;
BENJAPONG, W ;
DURIYANANDA, D ;
UNGKASRITHONGKUL, M .
TRANSACTIONS OF THE ROYAL SOCIETY OF TROPICAL MEDICINE AND HYGIENE, 1983, 77 (03) :338-340
[7]   ANALYSIS OF FILTER-PAPER-ABSORBED, FINGER-STICK BLOOD-SAMPLES FOR CHLOROQUINE AND ITS MAJOR METABOLITE USING HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHY WITH FLUORESCENCE DETECTION [J].
PATCHEN, LC ;
MOUNT, DL ;
SCHWARTZ, IK ;
CHURCHILL, FC .
JOURNAL OF CHROMATOGRAPHY, 1983, 278 (01) :81-89
[8]   DETERMINATION OF DRUG SENSITIVITY OF PLASMODIUM-FALCIPARUM [J].
RIECKMANN, KH .
JOURNAL OF THE AMERICAN MEDICAL ASSOCIATION, 1971, 217 (05) :573-+
[9]  
TRENHOLME GM, 1974, B WORLD HEALTH ORGAN, V51, P431
[10]  
WERNSDORFER WH, 1983, WHO CHRON, V37, P11