SYNTHESIS OF 5,6-METHYLENEDIOXY-1-TETRALONE - AN ARYL GRIGNARD APPROACH FROM GUAIACOL

被引：14

作者：

KLIX, RC

CAIN, MH

BHATIA, AV

机构：

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 36期

关键词：

D O I：

10.1016/0040-4039(95)01343-G

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A convenient synthesis of 5,6-methylenedioxy-1-tetralone (1) is described. The main features of this synthesis are the formation of 6 via a Grignard reaction using succinic anhydride followed by selective reduction and Friedel-Crafts cyclization to generate the desired tetralone 1.

引用

页码：6413 / 6414

页数：2

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