BEHAVIORAL AND RADIOLIGAND BINDING EVIDENCE FOR IRREVERSIBLE DOPAMINE RECEPTOR BLOCKADE BY N-ETHOXYCARBONYL-2-ETHOXY-1,2-DIHYDROQUINOLINE

被引：150

作者：

HAMBLIN, MW

CREESE, I

机构：

来源：

LIFE SCIENCES | 1983年 / 32卷 / 19期

关键词：

D O I：

10.1016/0024-3205(83)90423-X

中图分类号：

R-3 [医学研究方法]; R3 [基础医学];

学科分类号：

1001 ;

摘要：

引用

收藏

页码：2247 / 2255

页数：9

相关论文

共 22 条

[1] N-CARBOXYLIC ACID ESTERS OF 1,2- AND 1,4-DIHYDROQUINOLINES . A NEW CLASS OF IRREVERSIBLE INACTIVATORS OF CATECHOLAMINE ALPHA RECEPTORS AND POTENT CENTRAL NERVOUS SYSTEM DEPRESSANTS
BELLEAU, B
MARTEL, R
LACASSE, G
MENARD, M
WEINBERG, NL
PERRON, YG
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1968, 90 (03) : 823 - &
[2] MECHANISM OF IRREVERSIBLE ADRENERGIC BLOCKADE BY N-CARBETHOXYDIHYDROQUINOLINES - MODEL STUDIES WITH TYPICAL SERINE HYDROLASES
BELLEAU, B
DITULLIO, V
GODIN, D
[J]. BIOCHEMICAL PHARMACOLOGY, 1969, 18 (05) : 1039 - &
[3] A NEW CONVENIENT REAGENT FOR PEPTIDE SYNTHESES
BELLEAU, B
MALEK, G
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1968, 90 (06) : 1651 - &
[4] BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[5] Chang K., 1970, PHARMACOL RES COMMUN, V2, P63
[6] ON THE ABILITY OF N-CHLOROETHYL APORPHINE DERIVATIVES TO CAUSE IRREVERSIBLE INHIBITION OF DOPAMINE RECEPTOR MECHANISMS
COSTALL, B
FORTUNE, DH
GRANCHELLI, FE
LAW, SJ
NAYLOR, RJ
NEUMEYER, JL
NOHRIA, V
[J]. JOURNAL OF PHARMACY AND PHARMACOLOGY, 1980, 32 (08) : 571 - 576
[7] (-)N-(CHLOROETHYL)NORAPOMORPHINE INHIBITS STRIATAL DOPAMINE FUNCTION VIA IRREVERSIBLE RECEPTOR-BINDING
COSTALL, B
FORTUNE, DH
LAW, SJ
NAYLOR, RJ
NEUMEYER, JL
NOHRIA, V
[J]. NATURE, 1980, 285 (5766) : 571 - 573
[8] DOPAMINE RECEPTOR-BINDING PREDICTS CLINICAL AND PHARMACOLOGICAL POTENCIES OF ANTI-SCHIZOPHRENIC DRUGS
CREESE, I
BURT, DR
SNYDER, SH
[J]. SCIENCE, 1976, 192 (4238) : 481 - 483
[9] BLOCKAGE OF AMPHETAMINE INDUCED MOTOR STIMULATION AND STEREOTYPY IN ADULT RAT FOLLOWING NEONATAL TREATMENT WITH 6-HYDROXYDOPAMINE
CREESE, I
IVERSEN, SD
[J]. BRAIN RESEARCH, 1973, 55 (02) : 369 - 382
[10] CREESE I, 1978, NEUROTRANSMITTER REC, P141