N,N''-(DITHIO-2,1-ETHANEDIYL)BIS(N'-(PYRROL-2-YLMETHYL)-1,6-HEXANEDIAMINE)(PYREXTRAMINE), A NEW IRREVERSIBLE ALPHA-1-ADRENORECEPTOR BLOCKING-AGENT OF THE TETRAMINE DISULFIDE CLASS

被引：10

作者：

BRASILI, L ^{[1
]}

ANGELI, P ^{[1
]}

BRANCIA, E ^{[1
]}

MELCHIORRE, C ^{[1
]}

机构：

[1] UNIV CAMERINO,DEPT CHEM SCI,I-62032 CAMERINO,ITALY

来源：

EUROPEAN JOURNAL OF PHARMACOLOGY | 1984年 / 103卷 / 1-2期

关键词：

D O I：

10.1016/0014-2999(84)90209-7

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：181 / 184

页数：4

共 10 条

[1] IRREVERSIBLE ALPHA-ADRENOCEPTOR BLOCKING EFFECTS AND REVERSIBLE MUSCARINIC BLOCKING AND NICOTINIC BLOCKING EFFECTS OF TETRAMINE DISULFIDES ON THE HEART [J].

BENFEY, BG ;

BELLEAU, B ;

BRASILI, L ;

GIANNELLA, M ;

MELCHIORRE, C .

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1980, 58 (12) :1477-1483

[2] INHIBITION OF THE CARDIAC INOTROPIC EFFECT OF PHENYLEPHRINE BY A TETRAMINE DISULFIDE WITH IRREVERSIBLE ALPHA-ADRENOCEPTOR BLOCKING ACTIVITY [J].

BENFEY, BG ;

YONG, MS ;

BELLEAU, B ;

MELCHIORRE, C .

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1979, 57 (05) :510-516

[3]

BRAZENOR RM, 1981, J PHARMACOL EXP THER, V218, P530

[4] DEMONSTRATION OF ALPHA-1S-ADRENOCEPTORS AFTER EXPOSURE OF THE RAT ANOCOCCYGEUS TO BENEXTRAMINE [J].

COATES, J ;

WEETMAN, DF .

BRITISH JOURNAL OF PHARMACOLOGY, 1983, 80 (02) :343-346

[5]

FURCHGOTT RF, 1980, VASCULAR NEUROEFFECT, P245

[6]

KENAKIN TP, 1981, J PHARMACOL EXP THER, V216, P210

[7] TETRAMINE DISULFIDES - A NEW TOOL IN ALPHA-ADRENERGIC PHARMACOLOGY [J].

MELCHIORRE, C .

TRENDS IN PHARMACOLOGICAL SCIENCES, 1981, 2 (08) :209-211

[8]

MELCHIORRE C, 1983, FARMACO-ED SCI, V38, P950

[9] MOLECULAR-PROPERTIES OF ADRENERGIC ALPHA-RECEPTOR .2. OPTIMUM COVALENT INHIBITION BY 2 DIFFERENT PROTOTYPES OF POLYAMINE DISULFIDES [J].

MELCHIORRE, C ;

YONG, MS ;

BENFEY, BG ;

BELLEAU, B .

JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (11) :1126-1132

[10]

Tallarida R.J., 1979, DOSE RESPONSE RELATI

← 1 →