ACTIVITY OF QUINOLINE-CONTAINING ANTIMALARIALS AGAINST CHLOROQUINE-SENSITIVE AND CHLOROQUINE-RESISTANT STRAINS OF PLASMODIUM-FALCIPARUM INVITRO

被引:41
作者
GEARY, TG [1 ]
DIVO, AA [1 ]
JENSEN, JB [1 ]
机构
[1] MICHIGAN STATE UNIV, DEPT MICROBIOL & PUBL HLTH, E LANSING, MI 48824 USA
关键词
D O I
10.1016/0035-9203(87)90175-1
中图分类号
R1 [预防医学、卫生学];
学科分类号
1004 ; 120402 ;
摘要
引用
收藏
页码:499 / 503
页数:5
相关论文
共 23 条
[1]   INVITRO ASSESSMENT OF THE ANTIMALARIAL ACTIVITY OF CHLOROQUINE AND ITS MAJOR METABOLITES [J].
ADEROUNMU, AF .
ANNALS OF TROPICAL MEDICINE AND PARASITOLOGY, 1984, 78 (06) :581-585
[2]  
ADEROUNMU AF, 1983, J PHARMACOL EXP THER, V226, P633
[3]   HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC ANALYSIS OF THE METABOLISM OF PRIMAQUINE AND THE IDENTIFICATION OF A NEW MAMMALIAN METABOLITE [J].
BAKER, JK ;
MCCHESNEY, JD ;
HUFFORD, CD ;
CLARK, AM .
JOURNAL OF CHROMATOGRAPHY, 1982, 230 (01) :69-77
[4]   HIGH-AFFINITY BINDING OF QUININE TO IRON(III) PORPHYRINS - NOVEL FORMATION OF ALKOXIDE COMPLEXES FROM ALCOHOLS AND AMINES [J].
BEHERE, DV ;
GOFF, HM .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1984, 106 (17) :4945-4950
[5]   EVALUATION OF AMODIAQUINE TREATMENT OF CHLOROQUINE-RESISTANT PLASMODIUM-FALCIPARUM MALARIA ON ZANZIBAR, 1982 [J].
CAMPBELL, CC ;
PAYNE, D ;
SCHWARTZ, IK ;
KHATIB, OJ .
AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, 1983, 32 (06) :1216-1220
[6]   AMODIAQUINE AS A PRODRUG - IMPORTANCE OF METABOLITE(S) IN THE ANTIMALARIAL EFFECT OF AMODIAQUINE IN HUMANS [J].
CHURCHILL, FC ;
PATCHEN, LC ;
CAMPBELL, CC ;
SCHWARTZ, IK ;
PHUC, ND ;
DICKINSON, CM .
LIFE SCIENCES, 1985, 36 (01) :53-62
[7]   QUANTITATIVE ASSESSMENT OF ANTI-MALARIAL ACTIVITY INVITRO BY A SEMIAUTOMATED MICRODILUTION TECHNIQUE [J].
DESJARDINS, RE ;
CANFIELD, CJ ;
HAYNES, JD ;
CHULAY, JD .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1979, 16 (06) :710-718
[8]  
FITCH CD, 1972, P HELM SOC WASH, V39, P265
[9]  
FITCH CD, 1983, CIBA F SYMP, V94, P222
[10]   THE SINGLE DOSE KINETICS OF CHLOROQUINE AND ITS MAJOR METABOLITE DESETHYLCHLOROQUINE IN HEALTHY-SUBJECTS [J].
FRISKHOLMBERG, M ;
BERGQVIST, Y ;
TERMOND, E ;
DOMEIJNYBERG, B .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1984, 26 (04) :521-530