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NONPEPTIDE FIBRINOGEN RECEPTOR ANTAGONISTS .1. DISCOVERY AND DESIGN OF EXOSITE INHIBITORS
被引:276
作者
:
HARTMAN, GD
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
HARTMAN, GD
[
1
]
EGBERTSON, MS
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
EGBERTSON, MS
[
1
]
HALCZENKO, W
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
HALCZENKO, W
[
1
]
LASWELL, WL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
LASWELL, WL
[
1
]
DUGGAN, ME
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
DUGGAN, ME
[
1
]
SMITH, RL
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
SMITH, RL
[
1
]
NAYLOR, AM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
NAYLOR, AM
[
1
]
MANNO, PD
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MANNO, PD
[
1
]
LYNCH, RJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
LYNCH, RJ
[
1
]
ZHANG, GX
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
ZHANG, GX
[
1
]
CHANG, CTC
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
CHANG, CTC
[
1
]
GOULD, RJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
GOULD, RJ
[
1
]
机构
:
[1]
MERCK RES LABS,DEPT PHARMACOL,W POINT,PA 19486
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1992年
/ 35卷
/ 24期
关键词
:
D O I
:
10.1021/jm00102a020
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
[No abstract available]
引用
收藏
页码:4640 / 4642
页数:3
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IDENTIFICATION AND CHARACTERIZATION OF CELL-SUBSTRATUM ADHESION RECEPTORS ON CULTURED HUMAN-ENDOTHELIAL CELLS
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[J].
JOURNAL OF CLINICAL INVESTIGATION,
1989,
83
(06)
: 1992
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2002
[2]
EXPOSURE OF PLATELET FIBRINOGEN RECEPTORS BY ADP AND EPINEPHRINE
BENNETT, JS
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0
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VILAIRE, G
论文数:
0
引用数:
0
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[J].
JOURNAL OF CLINICAL INVESTIGATION,
1979,
64
(05)
: 1393
-
1401
[3]
A NEW MURINE MONOCLONAL-ANTIBODY REPORTS AN ACTIVATION-DEPENDENT CHANGE IN THE CONFORMATION AND OR MICROENVIRONMENT OF THE PLATELET GLYCOPROTEIN IIB/IIIA COMPLEX
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0
引用数:
0
h-index:
0
机构:
SUNY STONY BROOK, DIV HEMATOL, STONY BROOK, NY 11794 USA
SUNY STONY BROOK, DIV HEMATOL, STONY BROOK, NY 11794 USA
COLLER, BS
[J].
JOURNAL OF CLINICAL INVESTIGATION,
1985,
76
(01)
: 101
-
108
[4]
A MURINE MONOCLONAL-ANTIBODY THAT COMPLETELY BLOCKS THE BINDING OF FIBRINOGEN TO PLATELETS PRODUCES A THROMBASTHENIC-LIKE STATE IN NORMAL PLATELETS AND BINDS TO GLYCOPROTEINS-IIB AND OR GLYCOPROTEIN-IIIA
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h-index:
0
机构:
SUNY STONY BROOK, DEPT MICROBIOL, STONY BROOK, NY 11794 USA
COLLER, BS
PEERSCHKE, EI
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引用数:
0
h-index:
0
机构:
SUNY STONY BROOK, DEPT MICROBIOL, STONY BROOK, NY 11794 USA
PEERSCHKE, EI
SCUDDER, LE
论文数:
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SUNY STONY BROOK, DEPT MICROBIOL, STONY BROOK, NY 11794 USA
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72
(01)
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Colman RW, 1987, HEMOSTASIS THROMBOSI, P3
[6]
DAVIES MJ, 1985, BRIT HEART J, V53, P363
[7]
UNSTABLE ANGINA WITH FATAL OUTCOME - DYNAMIC CORONARY THROMBOSIS LEADING TO INFARCTION AND OR SUDDEN-DEATH - AUTOPSY EVIDENCE OF RECURRENT MURAL THROMBOSIS WITH PERIPHERAL EMBOLIZATION CULMINATING IN TOTAL VASCULAR OCCLUSION
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RANDERS CENT SYGEHUS,INST PATHOL,AALBORG,DENMARK
FALK, E
[J].
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71
(04)
: 699
-
708
[8]
PLATELET ACTIVATION IN UNSTABLE CORONARY-DISEASE
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[J].
NEW ENGLAND JOURNAL OF MEDICINE,
1986,
315
(16)
: 983
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989
[9]
GAN ZR, 1988, J BIOL CHEM, V263, P19827
[10]
CHEMICAL SYNTHESIS OF ECHISTATIN, A POTENT INHIBITOR OF PLATELET-AGGREGATION FROM ECHIS-CARINATUS - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SELECTED ANALOGS
GARSKY, VM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
GARSKY, VM
LUMMA, PK
论文数:
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引用数:
0
h-index:
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机构:
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MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
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FRIEDMAN, PA
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1989,
86
(11)
: 4022
-
4026
←
1
2
3
4
→
共 31 条
[1]
IDENTIFICATION AND CHARACTERIZATION OF CELL-SUBSTRATUM ADHESION RECEPTORS ON CULTURED HUMAN-ENDOTHELIAL CELLS
ALBELDA, SM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PENN,SCH MED,DEPT MED,DIV CARDIOVASC PULM,PHILADELPHIA,PA 19104
ALBELDA, SM
DAISE, M
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PENN,SCH MED,DEPT MED,DIV CARDIOVASC PULM,PHILADELPHIA,PA 19104
DAISE, M
LEVINE, EM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PENN,SCH MED,DEPT MED,DIV CARDIOVASC PULM,PHILADELPHIA,PA 19104
LEVINE, EM
BUCK, CA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV PENN,SCH MED,DEPT MED,DIV CARDIOVASC PULM,PHILADELPHIA,PA 19104
BUCK, CA
[J].
JOURNAL OF CLINICAL INVESTIGATION,
1989,
83
(06)
: 1992
-
2002
[2]
EXPOSURE OF PLATELET FIBRINOGEN RECEPTORS BY ADP AND EPINEPHRINE
BENNETT, JS
论文数:
0
引用数:
0
h-index:
0
BENNETT, JS
VILAIRE, G
论文数:
0
引用数:
0
h-index:
0
VILAIRE, G
[J].
JOURNAL OF CLINICAL INVESTIGATION,
1979,
64
(05)
: 1393
-
1401
[3]
A NEW MURINE MONOCLONAL-ANTIBODY REPORTS AN ACTIVATION-DEPENDENT CHANGE IN THE CONFORMATION AND OR MICROENVIRONMENT OF THE PLATELET GLYCOPROTEIN IIB/IIIA COMPLEX
COLLER, BS
论文数:
0
引用数:
0
h-index:
0
机构:
SUNY STONY BROOK, DIV HEMATOL, STONY BROOK, NY 11794 USA
SUNY STONY BROOK, DIV HEMATOL, STONY BROOK, NY 11794 USA
COLLER, BS
[J].
JOURNAL OF CLINICAL INVESTIGATION,
1985,
76
(01)
: 101
-
108
[4]
A MURINE MONOCLONAL-ANTIBODY THAT COMPLETELY BLOCKS THE BINDING OF FIBRINOGEN TO PLATELETS PRODUCES A THROMBASTHENIC-LIKE STATE IN NORMAL PLATELETS AND BINDS TO GLYCOPROTEINS-IIB AND OR GLYCOPROTEIN-IIIA
COLLER, BS
论文数:
0
引用数:
0
h-index:
0
机构:
SUNY STONY BROOK, DEPT MICROBIOL, STONY BROOK, NY 11794 USA
COLLER, BS
PEERSCHKE, EI
论文数:
0
引用数:
0
h-index:
0
机构:
SUNY STONY BROOK, DEPT MICROBIOL, STONY BROOK, NY 11794 USA
PEERSCHKE, EI
SCUDDER, LE
论文数:
0
引用数:
0
h-index:
0
机构:
SUNY STONY BROOK, DEPT MICROBIOL, STONY BROOK, NY 11794 USA
SCUDDER, LE
SULLIVAN, CA
论文数:
0
引用数:
0
h-index:
0
机构:
SUNY STONY BROOK, DEPT MICROBIOL, STONY BROOK, NY 11794 USA
SULLIVAN, CA
[J].
JOURNAL OF CLINICAL INVESTIGATION,
1983,
72
(01)
: 325
-
338
[5]
Colman RW, 1987, HEMOSTASIS THROMBOSI, P3
[6]
DAVIES MJ, 1985, BRIT HEART J, V53, P363
[7]
UNSTABLE ANGINA WITH FATAL OUTCOME - DYNAMIC CORONARY THROMBOSIS LEADING TO INFARCTION AND OR SUDDEN-DEATH - AUTOPSY EVIDENCE OF RECURRENT MURAL THROMBOSIS WITH PERIPHERAL EMBOLIZATION CULMINATING IN TOTAL VASCULAR OCCLUSION
FALK, E
论文数:
0
引用数:
0
h-index:
0
机构:
RANDERS CENT SYGEHUS,INST PATHOL,AALBORG,DENMARK
RANDERS CENT SYGEHUS,INST PATHOL,AALBORG,DENMARK
FALK, E
[J].
CIRCULATION,
1985,
71
(04)
: 699
-
708
[8]
PLATELET ACTIVATION IN UNSTABLE CORONARY-DISEASE
FITZGERALD, DJ
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,DIV CARDIOL,NASHVILLE,TN 37232
FITZGERALD, DJ
ROY, L
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,DIV CARDIOL,NASHVILLE,TN 37232
ROY, L
CATELLA, F
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,DIV CARDIOL,NASHVILLE,TN 37232
CATELLA, F
FITZGERALD, GA
论文数:
0
引用数:
0
h-index:
0
机构:
VANDERBILT UNIV,DIV CARDIOL,NASHVILLE,TN 37232
FITZGERALD, GA
[J].
NEW ENGLAND JOURNAL OF MEDICINE,
1986,
315
(16)
: 983
-
989
[9]
GAN ZR, 1988, J BIOL CHEM, V263, P19827
[10]
CHEMICAL SYNTHESIS OF ECHISTATIN, A POTENT INHIBITOR OF PLATELET-AGGREGATION FROM ECHIS-CARINATUS - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF SELECTED ANALOGS
GARSKY, VM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
GARSKY, VM
LUMMA, PK
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
LUMMA, PK
FREIDINGER, RM
论文数:
0
引用数:
0
h-index:
0
机构:
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MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
FREIDINGER, RM
PITZENBERGER, SM
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
PITZENBERGER, SM
RANDALL, WC
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
RANDALL, WC
VEBER, DF
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
VEBER, DF
GOULD, RJ
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
GOULD, RJ
FRIEDMAN, PA
论文数:
0
引用数:
0
h-index:
0
机构:
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
MERCK SHARP & DOHME RES LABS,DEPT PHARMACOL,W POINT,PA 19486
FRIEDMAN, PA
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1989,
86
(11)
: 4022
-
4026
←
1
2
3
4
→