A DIRECT PREPARATION OF 1,4-BENZODIAZEPINES - THE SYNTHESIS OF MEDAZEPAM AND RELATED-COMPOUNDS VIA A COMMON INTERMEDIATE

被引：26

作者：

KRAUS, GA

MAEDA, H

机构：

[1] Department of Chemistry, Iowa State University, Ames

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 49期

关键词：

BENZODIAZEPINE; TRIFLATE; PALLADIUM; PHOTOCHEMISTRY;

D O I：

10.1016/0040-4039(94)88461-7

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The benzodiazepine skeleton was prepared from benzoquinone in three steps. Medazepam was prepared from 9.

引用

页码：9189 / 9190

页数：2

共 9 条

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[3]

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[4]

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[6]

KRAUS GA, 1994, IN PRESS ACS MONOGRA

[7]

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[8]

ROTH HJ, 1987, PHARM CHEM, V1

[9] QUINAZOLINES AND BENZODIAZEPINES .15. 7-NITRO- AND 7-TRIFLUOROMETHYL-2,3-DIHYDRO-5-PHENYL-1H-1,4-BENZODIAZEPINES AND THEIR TRANSFORMATIONS [J].

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ARCHER, GA ;

REEDER, E .

JOURNAL OF ORGANIC CHEMISTRY, 1963, 28 (11) :3013-&

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