USE-DEPENDENT BLOCK OF CARDIAC SODIUM-CHANNELS BY QUATERNARY DERIVATIVES OF LIDOCAINE

被引:22
作者
GINTANT, GA
HOFFMAN, BF
机构
[1] COLUMBIA UNIV COLL PHYS & SURG,DEPT PHARMACOL,NEW YORK,NY 10032
[2] SUNY STONY BROOK,HLTH SCI CTR,DEPT PHYSIOL & BIOPHYS,STONY BROOK,NY 11794
来源
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY | 1984年 / 400卷 / 02期
关键词
D O I
10.1007/BF00585029
中图分类号
Q4 [生理学];
学科分类号
071003 ;
摘要
引用
收藏
页码:121 / 129
页数:9
相关论文
共 52 条
[1]   STEADY-STATE TTX-SENSITIVE (WINDOW) SODIUM CURRENT IN CARDIAC PURKINJE-FIBERS [J].
ATTWELL, D ;
COHEN, I ;
EISNER, D ;
OHBA, M ;
OJEDA, C .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1979, 379 (02) :137-142
[2]   SODIUM-CHANNEL INACTIVATION IN THE CRAYFISH GIANT-AXON - MUST CHANNELS OPEN BEFORE INACTIVATING [J].
BEAN, BP .
BIOPHYSICAL JOURNAL, 1981, 35 (03) :595-614
[3]  
BEAN BP, 1982, NORMAL ABNORMAL COND
[4]  
BIGGER JT, 1980, PHARMACOL BASIS THER, P761
[5]  
BROWN AM, 1981, J PHYSIOL-LONDON, V318, P479
[6]   LOCAL-ANESTHETIC BLOCK OF SODIUM CHANNELS IN NORMAL AND PRONASE-TREATED SQUID GIANT-AXONS [J].
CAHALAN, MD .
BIOPHYSICAL JOURNAL, 1978, 23 (02) :285-311
[7]   SHORTENING OF THE ACTION-POTENTIAL AND REDUCTION OF PACEMAKER ACTIVITY BY LIDOCAINE, QUINIDINE, AND PROCAINAMIDE IN SHEEP CARDIAC PURKINJE-FIBERS - AN EFFECT ON NA OR K CURRENTS [J].
CARMELIET, E ;
SAIKAWA, T .
CIRCULATION RESEARCH, 1982, 50 (02) :257-272
[8]   EFFECT OF LIDOCAINE AND QUINIDINE ON STEADY-STATE CHARACTERISTICS AND RECOVERY KINETICS OF (DV-DT) MAX IN GUINEA-PIG VENTRICULAR MYOCARDIUM [J].
CHEN, CM ;
GETTES, LS ;
KATZUNG, BG .
CIRCULATION RESEARCH, 1975, 37 (01) :20-29
[9]   TETRODOTOXIN BLOCK OF SODIUM-CHANNELS IN RABBIT PURKINJE-FIBERS - INTERACTIONS BETWEEN TOXIN BINDING AND CHANNEL GATING [J].
COHEN, CJ ;
BEAN, BP ;
COLATSKY, TJ ;
TSIEN, RW .
JOURNAL OF GENERAL PHYSIOLOGY, 1981, 78 (04) :383-411
[10]   THE DEPENDENCE OF THE MAXIMUM RATE OF RISE OF THE ACTION-POTENTIAL UPSTROKE ON MEMBRANE-PROPERTIES [J].
COHEN, I ;
ATTWELL, D ;
STRICHARTZ, G .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1981, 214 (1194) :85-98