QUINAZOLINE ANTIFOLATES INHIBITING THYMIDYLATE SYNTHASE - 2-DESAMINO DERIVATIVES WITH ENHANCED SOLUBILITY AND POTENCY

被引：80

作者：

JONES, TR ^{[1
]}

THORNTON, TJ ^{[1
]}

FLINN, A ^{[1
]}

JACKMAN, AL ^{[1
]}

NEWELL, DR ^{[1
]}

CALVERT, AH ^{[1
]}

机构：

[1] INST CANC RES, DRUG DEV SECT, SUTTON SM2 5NG, SURREY, ENGLAND

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1989年 / 32卷 / 04期

关键词：

D O I：

10.1021/jm00124a018

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：847 / 852

页数：6

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