ABSENCE OF [H-3] SCH-23390 SPECIFIC BINDING-SITES IN ANTERIOR-PITUITARY - DISSOCIATION FROM EFFECTS ON PROLACTIN SECRETION

被引:20
作者
ROVESCALLI, AC
BRUNELLO, N
MONOPOLI, A
ONGINI, E
RACAGNI, G
机构
[1] ESSEX ITALIA COMAZZO,RES LABS,MILANO,ITALY
[2] UNIV PAVIA,INST PHARMACOL,I-27100 PAVIA,ITALY
关键词
D O I
10.1016/0014-2999(87)90604-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:129 / 136
页数:8
相关论文
共 26 条
[1]   INTERACTION OF SCH-23390, A D-1-SELECTIVE ANTAGONIST, WITH THE ANTERIOR-PITUITARY D-2 RECEPTORS AND PROLACTIN SECRETION IN THE RAT [J].
APUD, JA ;
MASOTTO, C ;
ONGINI, E ;
RACAGNI, G .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 112 (02) :187-193
[2]  
BARNETT A, 1986, Drugs of the Future, V11, P49
[3]   CHARACTERIZATION OF THE BINDING OF H-3-SCH 23390, A SELECTIVE D-1 RECEPTOR ANTAGONIST LIGAND, IN RAT STRIATUM [J].
BILLARD, W ;
RUPERTO, V ;
CROSBY, G ;
IORIO, LC ;
BARNETT, A .
LIFE SCIENCES, 1984, 35 (18) :1885-1893
[4]   PREFERENTIAL INHIBITION OF LIGAND-BINDING TO CALF STRIATAL DOPAMINE D1-RECEPTORS BY SCH-23390 [J].
CROSS, AJ ;
MASHAL, RD ;
JOHNSON, JA ;
OWEN, F .
NEUROPHARMACOLOGY, 1983, 22 (11) :1327-1329
[5]  
del Pozo E, 1979, Horm Res, V10, P143, DOI 10.1159/000178998
[6]   THE BENZAZEPINE SCH-23390 INCREASES PLASMA-LEVELS OF CORTISOL IN THE CONSCIOUS DOG [J].
GOINY, M ;
HERRERAMARSCHITZ, M ;
UVNASMOBERG, K ;
CEKAN, S ;
UNGERSTEDT, U .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1986, 332 (01) :111-112
[7]   SCH-23390 - THE 1ST SELECTIVE DOPAMINE D-1 ANTAGONIST [J].
HYTTEL, J .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 91 (01) :153-154
[8]  
IORIO LC, 1983, J PHARMACOL EXP THER, V226, P462
[9]   THE D-1 DOPAMINE RECEPTOR - NEW PERSPECTIVES [J].
KEBABIAN, JW ;
AGUI, T ;
VANOENE, JC ;
SHIGEMATSU, K ;
SAAVEDRA, JM .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1986, 7 (03) :96-99
[10]   ON THE MODE OF THE PROLACTIN RELEASE-INHIBITING ACTION OF THE SEROTONIN RECEPTOR BLOCKERS METERGOLINE, METHYSERGIDE, AND CYPROHEPTADINE [J].
KRULICH, L ;
MCCANN, SM ;
MAYFIELD, MA .
ENDOCRINOLOGY, 1981, 108 (04) :1115-1124