HUMAN PHARMACOKINETICS OF TEMOCILLIN (BRL-17421) SIDE-CHAIN EPIMERS

被引:8
作者
GUEST, EA [1 ]
HORTON, R [1 ]
MELLOWS, G [1 ]
SLOCOMBE, B [1 ]
SWAISLAND, AJ [1 ]
TASKER, TCG [1 ]
机构
[1] BIOSCI RES CTR,EPSOM,SURREY,ENGLAND
关键词
D O I
10.1093/jac/15.3.327
中图分类号
R51 [传染病];
学科分类号
100401 ;
摘要
引用
收藏
页码:327 / 336
页数:10
相关论文
共 13 条
[1]   HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC ASSAY OF TEMOCILLIN AND EPIMERIZATION OF ITS DIASTEREOISOMERS [J].
BIRD, AE ;
CHARSLEY, CH ;
JENNINGS, KR ;
MARSHALL, AC .
ANALYST, 1984, 109 (09) :1209-1212
[2]   TEMOCILLIN, INVITRO ACTIVITY AND THE PHARMACOKINETICS AND TISSUE PENETRATION IN HEALTHY-VOLUNTEERS [J].
BROWN, RM ;
WISE, R ;
ANDREWS, JM .
JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY, 1982, 10 (04) :295-302
[3]  
GIBALDI M, 1975, PHARMACOKINETICS
[4]   SEPARATION OF THE SIDE-CHAIN DIASTEREOISOMERS OF PENICILLINS BY HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHY [J].
HOOGMARTENS, J ;
ROETS, E ;
JANSSEN, G ;
VANDERHAEGHE, H .
JOURNAL OF CHROMATOGRAPHY, 1982, 244 (02) :299-309
[5]  
JACKSON D, 1982, 12TH P ICC FLOR, P326
[6]   MOXALACTAM EPIMER KINETICS IN CHILDREN [J].
NAHATA, MC ;
DURRELL, DE ;
BARSON, WJ .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1982, 31 (04) :528-532
[7]   RENAL EXCRETION OF R-EPIMERS AND S-EPIMERS OF MOXALACTAM IN DOGS [J].
NAKAMURA, M ;
SUGENO, K ;
KONAKA, R ;
YAMADA, H ;
YOSHIDA, T .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1982, 71 (10) :1188-1189
[8]   BRL-17421, A NOVEL BETA-LACTAM ANTIBIOTIC, HIGHLY RESISTANT TO BETA-LACTAMASES, GIVING HIGH AND PROLONGED SERUM LEVELS IN HUMANS [J].
SLOCOMBE, B ;
BASKER, MJ ;
BENTLEY, PH ;
CLAYTON, JP ;
COLE, M ;
COMBER, KR ;
DIXON, RA ;
EDMONDSON, RA ;
JACKSON, D ;
MERRIKIN, DJ ;
SUTHERLAND, R .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1981, 20 (01) :38-46
[10]  
WISE R, 1982, REV INFECT DIS, V4, pS564