SYNTHESIS OF 3'-C-CYANO-3'-DEOXY-PENTOFURANOSYLTHYMINE NUCLEOSIDES

被引：33

作者：

CALVOMATEO, A

CAMARASA, MJ

DIAZORTIZ, A

HERAS, FGD

ALEMANY, A

机构：

[1] INST QUIM MED,JUAN CIERVA 3,E-28006 MADRID,SPAIN

[2] INST QUIM ORGAN GEN,E-28006 MADRID,SPAIN

来源：

TETRAHEDRON | 1988年 / 44卷 / 15期

关键词：

D O I：

10.1016/S0040-4020(01)86194-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：4895 / 4903

页数：9

共 22 条

[1] THE SYNTHESIS OF SOME BRANCHED-CHAIN-SUGAR NUCLEOSIDE ANALOGS [J].

ASHWELL, M ;

JONES, AS ;

WALKER, RT .

NUCLEIC ACIDS RESEARCH, 1987, 15 (05) :2157-2166

[2] A GENERAL-METHOD FOR DETERMINING THE ANOMERIC CONFIGURATION OF C-FURANOSIDE DERIVATIVES - A H-1 NUCLEAR-MAGNETIC-RESONANCE NUCLEAR OVERHAUSER EFFECT STUDY [J].

BERNSTEIN, MA ;

MORTON, HE ;

GUINDON, Y .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 2, 1986, (08) :1155-1163

[3] 3'-C-CYANO-3'-DEOXYTHYMIDINE [J].

CALVOMATEO, A ;

CAMARASA, MJ ;

DIAZORTIZ, A ;

DELASHERAS, FG .

TETRAHEDRON LETTERS, 1988, 29 (08) :941-944

[4]

CALVOMATEO A, IN PRESS J CHEM SOC

[5]

DECLERCQ E, 1987, TRENDS PHARMACOL SCI, V8, P339

[6] CHEMOTHERAPEUTIC APPROACHES TO THE TREATMENT OF THE ACQUIRED-IMMUNE-DEFICIENCY-SYNDROME (AIDS) [J].

DECLERCQ, E .

JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (09) :1561-1569

[7] THE EFFICACY OF AZIDOTHYMIDINE (AZT) IN THE TREATMENT OF PATIENTS WITH AIDS AND AIDS-RELATED COMPLEX - A DOUBLE-BLIND, PLACEBO-CONTROLLED TRIAL [J].

FISCHL, MA ;

RICHMAN, DD ;

GRIECO, MH ;

GOTTLIEB, MS ;

VOLBERDING, PA ;

LASKIN, OL ;

LEEDOM, JM ;

GROOPMAN, JE ;

MILDVAN, D ;

SCHOOLEY, RT ;

JACKSON, GG ;

DURACK, DT ;

KING, D .

NEW ENGLAND JOURNAL OF MEDICINE, 1987, 317 (04) :185-191

[8] METHYL 5-O-TERT-BUTYLDIPHENYLSILYL-2-DEOXY-ALPHA,BETA-D-THREO-PENTOFURANOSIDE AS A DIVERGENT INTERMEDIATE FOR THE SYNTHESIS OF 3'-SUBSTITUTED-2',3'-DIDEOXYNUCLEOSIDES - SYNTHESIS OF 3'-AZIDO-3'-DEOXYTHYMIDINE, 3'-DEOXY-3'-FLUOROTHYMIDINE AND 3'-CYANO-3'-DEOXYTHYMIDINE [J].

FLEET, GWJ ;

SON, JC ;

DEROME, AE .

TETRAHEDRON, 1988, 44 (02) :625-636

[9]

FURUKAWA Y, 1970, CHEM PHARM BULL, V18, P554

[10] NUCLEIC-ACID RELATED-COMPOUNDS .44. 2' AND 3'-KETONUCLEOSIDES AND THEIR ARABINO AND XYLO REDUCTION PRODUCTS - CONVENIENT ACCESS VIA SELECTIVE PROTECTION AND OXIDATION OF RIBONUCLEOSIDES [J].

HANSSKE, F ;

MADEJ, D ;

ROBINS, MJ .

TETRAHEDRON, 1984, 40 (01) :125-135

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