COMPARATIVE PHARMACOKINETIC STUDIES OF TIXOCORTOL PIVALATE AND CORTISOL IN THE RAT

被引:16
作者
CHANOINE, F
JUNIEN, JL
机构
关键词
D O I
10.1016/0022-4731(84)90311-X
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:453 / 459
页数:7
相关论文
共 19 条
[1]   UPTAKE OF CORTISOL BY RAT TISSUES [J].
BELLAMY, D ;
PHILLIPS, JG ;
CHESTERJ.I ;
LEONARD, RA .
BIOCHEMICAL JOURNAL, 1962, 85 (03) :537-&
[2]  
CHU NI, 1979, DRUG METAB DISPOS, V7, P81
[3]  
DAVIES JE, 1981, ARZNEIMITTEL-FORSCH, V31-1, P453
[4]   DISTRIBUTION OF INJECTED CORTISOL-4-C-14 IN NORMAL AND SHOCKED RATS [J].
FIRSCHEIN, HE ;
DEVENUTO, F ;
FITCH, WM ;
PEARCE, EM ;
WESTPHAL, U .
ENDOCRINOLOGY, 1957, 60 (03) :347-358
[5]  
FLORINI JR, 1961, J PHARMACOL EXP THER, V131, P287
[6]  
GOMENI R, 1983, MEDINFO 83, P1022
[7]  
GULYASSY P, 1958, P SOC EXP BIOL MED, V98, P711
[8]  
HYDE PM, 1957, J BIOL CHEM, V227, P1063
[9]   TIXOCORTOL PIVALATE, A CORTICOSTEROID WITH NO SYSTEMIC GLUCOCORTICOID EFFECT AFTER ORAL, INTRARECTAL, AND INTRANASAL APPLICATION [J].
LAROCHELLE, P ;
DUSOUICH, P ;
BOLTE, E ;
LELORIER, J ;
GOYER, R .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1983, 33 (03) :343-350
[10]   AFFINITY OF TIXOCORTOL PIVALATE (JO-1016), TIXOCORTOL, CORTISOL ACETATE AND CORTISOL FOR DEXAMETHASONE RECEPTORS OF MOUSE THYMUS-CELLS AND RAT RENOMEDULLARY INTERSTITIAL-CELLS IN CULTURE - CORRELATION WITH THEIR BIOLOGICAL-ACTIVITIES [J].
LELIEVRE, V ;
JUNIEN, JL ;
GOYER, R ;
RUSSOMARIE, F .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1984, 20 (01) :363-366