A NEW, PALLADIUM-CATALYZED SYNTHESIS OF AROMATIC MERCAPTURIC ACID-DERIVATIVES

被引：83

作者：

CIATTINI, PG

MORERA, E

ORTAR, G

机构：

[1] UNIV ROMA LA SAPIENZA,DIPARTIMENTO STUDI FARMACEUT,I-00185 ROME,ITALY

[2] UNIV ROMA LA SAPIENZA,CNR,CTR STUDIO CHIM FARMACO,I-00185 ROME,ITALY

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 23期

关键词：

D O I：

10.1016/0040-4039(95)00677-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

N-Acetyl-L-cysteine methyl ester (1) reacts under mild conditions with aryl iodides 2 in the presence of a palladium catalyst prepared in situ from Pd(2)dba(3) and dppf to give S-aryl derivatives 3 in moderate to good yields.

引用

页码：4133 / 4136

页数：4

共 34 条

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