SYNTHESIS AND CHARACTERIZATION OF ALKYL-SUBSTITUTED, ALKENYL-SUBSTITUTED, ACYL-SUBSTITUTED AND NITROGEN-SUBSTITUTED DERIVATIVES OF THE POTENT PHOTOTOXIN ALPHA-TERTHIOPHENE

被引：31

作者：

SOUCYBREAU, C ^{[1
]}

MACEACHERN, A ^{[1
]}

LEITCH, LC ^{[1
]}

ARNASON, T ^{[1
]}

MORAND, P ^{[1
]}

机构：

[1] UNIV OTTAWA, OTTAWA CARLETON INST BIOL, OTTAWA K1N 6N5, ONTARIO, CANADA

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1991年 / 28卷 / 02期

关键词：

D O I：

10.1002/jhet.5570280239

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Some alkyl-, alkenyl-, acyl- and nitrogen- derivatives of alpha-terthienyl 1 have been synthesized in an effort to expand the potential insecticidal activity profile of this compound. The introduction of substituents was carried out directly on the alpha-terthienyl molecule. Three compounds were isolated in the nitration reaction and the compounds have been identified as 5-nitro-2,2':5',2''-terthiophene 5, 3'-nitro-2,2':5',2''-terthiophene 6 and 3-nitro-2,2':5',2''-terthiophene 7 respectively. Preliminary results of biological activity are reported.

引用

页码：411 / 416

页数：6

共 15 条

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