IMPLICATIONS OF STEREOSELECTIVITY IN RADIOLIGAND BINDING-STUDIES

被引:11
作者
HOYER, D
机构
关键词
D O I
10.1016/0165-6147(86)90328-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:227 / 230
页数:4
相关论文
共 21 条
[1]   (-)-S-[H-3]CGP-12177 AND ITS USE TO DETERMINE THE RATE CONSTANTS OF UNLABELED BETA-ADRENERGIC ANTAGONISTS [J].
AFFOLTER, H ;
HERTEL, C ;
JAEGGI, K ;
PORTENIER, M ;
STAEHELIN, M .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (03) :925-929
[2]  
BENNETT JP, 1978, NEUROTRANSMITTER REC, P57
[3]   THE ALPHA-ADRENOCEPTOR AND BETA-ADRENOCEPTOR BLOCKING POTENCIES OF LABETALOL AND ITS INDIVIDUAL STEREOISOMERS IN ANESTHETIZED DOGS AND IN ISOLATED-TISSUES [J].
BRITTAIN, RT ;
DREW, GM ;
LEVY, GP .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 77 (01) :105-114
[4]  
BURGISSER E, 1981, MOL PHARMACOL, V19, P205
[5]  
BURGISSER E, 1981, MOL PHARMACOL, V19, P509
[6]   [BE-2254-I-125, A NEW HIGH-AFFINITY RADIOLIGAND FOR ALPHA-1-ADRENOCEPTORS [J].
ENGEL, G ;
HOYER, D .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 73 (2-3) :221-224
[7]   [IODO-125]BE 2254, A NEW RADIOLIGAND FOR ALPHA-1-ADRENOCEPTORS [J].
ENGEL, G ;
HOYER, D .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1982, 4 :S25-S29
[8]   THE OPTICAL ISOMERS OF THE 1,4-DIHYDROPYRIDINE BAY K-8644 SHOW OPPOSITE EFFECTS ON CA CHANNELS [J].
FRANCKOWIAK, G ;
BECHEM, M ;
SCHRAMM, M ;
THOMAS, G .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 114 (02) :223-226
[9]   [I-125]-HEAT - 50-PERCENT OF THE LIGAND CAN BIND TO THE ALPHA-1-ADRENOCEPTORS WITH EXTREMELY HIGH-AFFINITY [J].
GLOSSMANN, H ;
LUBBECKE, F ;
HABERMANN, B .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 321 (01) :7-10
[10]   CENTRAL DOPAMINE RECEPTOR AGONIST AND ANTAGONIST ACTIONS OF THE ENANTIOMERS OF 3-PPP [J].
HJORTH, S ;
CARLSSON, A ;
CLARK, D ;
SVENSSON, K ;
WIKSTROM, H ;
SANCHEZ, D ;
LINDBERG, P ;
HACKSELL, U ;
ARVIDSSON, LE ;
JOHANSSON, A ;
NILSSON, JLG .
PSYCHOPHARMACOLOGY, 1983, 81 (02) :89-99