SYNTHESIS AND EVALUATION OF 1- AND 2-SUBSTITUTED FENTANYL ANALOGS FOR OPIOID ACTIVITY

被引：23

作者：

ESSAWI, MYH ^{[1
]}

PORTOGHESE, PS ^{[1
]}

机构：

[1] UNIV MINNESOTA,COLL PHARM,DEPT MED CHEM,MINNEAPOLIS,MN 55455

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1983年 / 26卷 / 03期

关键词：

D O I：

10.1021/jm00357a007

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：348 / 352

页数：5

共 21 条

[1] A REINVESTIGATION OF MIXED CARBONIC ANHYDRIDE METHOD OF PEPTIDE SYNTHESIS [J].

ANDERSON, GW ;

ZIMMERMAN, JE ;

CALLAHAN, FM .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1967, 89 (19) :5012-+

[2] CYANOHYDRIDOBORATE ANION AS A SELECTIVE REDUCING AGENT [J].

BORCH, RF ;

BERNSTEIN, MD ;

DURST, HD .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1971, 93 (12) :2897-+

[3] OPIATE RECEPTOR-BINDING AFFECTED DIFFERENTIALLY BY OPIATES AND OPIOID PEPTIDES [J].

CHILDERS, SR ;

CREESE, I ;

SNOWMAN, AM ;

SNYDER, SH .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 55 (01) :11-18

[4]

ESSAWI MYH, J ORG CHEM

[5] OPIATE RECEPTOR - MODEL EXPLAINING STRUCTURE-ACTIVITY-RELATIONSHIPS OF OPIATE AGONISTS AND ANTAGONISTS [J].

FEINBERG, AP ;

CREESE, I ;

SNYDER, SH .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1976, 73 (11) :4215-4219

[6] NOVEL ANALOGS OF ENKEPHALIN - IDENTIFICATION OF FUNCTIONAL-GROUPS REQUIRED FOR BIOLOGICAL-ACTIVITY [J].

GORIN, FA ;

BALASUBRAMANIAN, TM ;

CICERO, TJ ;

SCHWIETZER, J ;

MARSHALL, GR .

JOURNAL OF MEDICINAL CHEMISTRY, 1980, 23 (10) :1113-1122

[7] EFFECT OF MORPHINE ON ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS ASSESSMENT OF AGONIST AND ANTAGONIST POTENCIES OF NARCOTIC ANALGESICS [J].

HUGHES, J ;

KOSTERLITZ, HW ;

LESLIE, FM .

BRITISH JOURNAL OF PHARMACOLOGY, 1975, 53 (03) :371-381

[8]

Janssen P. A. J., 1964, U. S. Patent, Patent No. 3141823

[9] KINETIC PARAMETERS OF NARCOTIC AGONISTS AND ANTAGONISTS WITH PARTICULAR REFERENCE TO N-ALLYLNOROXYMORPHONE (NALOXONE) [J].

KOSTERLITZ, HW ;

WATT, AJ .

BRITISH JOURNAL OF PHARMACOLOGY, 1968, 33 (02) :266-+

[10]

LOBBEZOO MW, 1980, EUR J MED CHEM, V15, P357

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