FURTHER INVITRO AND INVIVO STUDIES WITH THE PUTATIVE PRESYNAPTIC DOPAMINE AGONIST N,N-DIPROPYL-7-HYDROXY-2-AMINOTETRALIN

被引:24
作者
MULDER, TBA [1 ]
DEVRIES, JB [1 ]
DIJKSTRA, D [1 ]
WIECHERS, JW [1 ]
GROL, CJ [1 ]
HORN, AS [1 ]
机构
[1] STATE UNIV GRONINGEN,DEPT MED CHEM,PHARMACEUT LAB,ANT DEUSINGLAAN 2,9713 AW GRONINGEN,NETHERLANDS
关键词
D O I
10.1007/BF00169305
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:494 / 501
页数:8
相关论文
共 56 条
[21]  
HOLZ RW, 1974, MOL PHARMACOL, V10, P746
[22]   RELATIONSHIP BETWEEN LEVELS AND UPTAKE OF SEROTONIN AND HIGH-AFFINITY [H-3]IMIPRAMINE RECOGNITION SITES IN THE RAT-BRAIN [J].
HRDINA, PD ;
PAPPAS, BA ;
ROBERTS, DCS ;
BIALIK, RJ ;
RYAN, CL .
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1985, 63 (10) :1239-1244
[23]   FUNCTIONAL EVIDENCE FOR SELECTIVE DOPAMINE D-1 RECEPTOR BLOCKADE BY SCH-23390 [J].
HYTTEL, J .
NEUROPHARMACOLOGY, 1984, 23 (12A) :1395-1401
[24]  
IMPERATO A, 1985, J NEUROSCI, V5, P297
[25]   NOVEL DOPAMINE RECEPTOR AGONISTS AND ANTAGONISTS WITH PREFERENTIAL ACTION ON AUTORECEPTORS [J].
JOHANSSON, AM ;
ARVIDSSON, LE ;
HACKSELL, U ;
NILSSON, JLG ;
SVENSSON, K ;
HJORTH, S ;
CLARK, D ;
CARLSSON, A ;
SANCHEZ, D ;
ANDERSSON, B ;
WIKSTROM, H .
JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (08) :1049-1053
[26]  
Konig JFR, 1963, RAT BRAIN STEREOTAXI, P162
[28]  
LANGER SZ, 1982, J PHARMACOL EXP THER, V222, P220
[29]   PSYCHOTOMIMETIC OPIATE RECEPTORS LABELED AND VISUALIZED WITH (+)-[H-3]3-(3-HYDROXYPHENYL)-N-(1-PROPYL)PIPERIDINE [J].
LARGENT, BL ;
GUNDLACH, AL ;
SNYDER, SH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1984, 81 (15) :4983-4987
[30]   CHARACTERIZATION OF DOPAMINE AUTORECEPTOR AND [H-3]-LABELED SPIPERONE BINDING-SITES INVITRO WITH CLASSICAL AND NOVEL DOPAMINE RECEPTOR AGONISTS [J].
LEHMANN, J ;
BRILEY, M ;
LANGER, SZ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 88 (01) :11-26