SYNTHETIC THYROTROPIN-RELEASING FACTOR ANALOGS .3. EFFECT OF REPLACEMENT OR MODIFICATION OF HISTIDINE RESIDUE ON BIOLOGICAL-ACTIVITY

被引：80

作者：

RIVIER, J

BURGUS, R

VALE, W

LING, N

MONAHAN, M

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1972年 / 15卷 / 05期

关键词：

D O I：

10.1021/jm00275a010

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：479 / &

共 23 条

[1] PEPTIDE SEQUENCING BY LOW RESOLUTION MASS SPECTROMETRY .I. USE OF ACETYLACETONYL DERIVATIVES TO IDENTIFY N-TERMINAL RESIDUES [J].

BACON, V ;

JELLUM, E ;

PATTON, W ;

PEREIRA, W ;

HALPERN, B .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1969, 37 (06) :878-&

[2] ACTIVITY-STRUCTURE RELATIONSHIPS OF THYROTROPIN RELEASING HORMONE [J].

BOWERS, CY ;

SIEVERTSSON, H ;

ENZMANN, F ;

FOLKERS, K .

BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1970, 40 (03) :683-+

[3] BIOLOGICAL ACTIVITY OF SYNTHETIC POLYPEPTIDE DERIVATIVES RELATED TO STRUCTURE OF HYPOTHALAMIC TRF [J].

BURGUS, R ;

DUNN, TF ;

DESIDERIO, DM ;

WARD, DN ;

VALE, W ;

GUILLEMIN, R ;

FELIX, AM ;

GILLESSEN, D ;

STUDER, RO .

ENDOCRINOLOGY, 1970, 86 (03) :573-+

[4]

CHANG JK, 1971, J MED CHEM, V14, P484

[5]

EDSALL JT, 1943, PROTEINS AMINO ACIDS, P85

[6]

FISCHER E, 1908, J LIEBIGS ANN CHEM, V363, P107

[7]

GIBIAN H, 1961, LIEBIGS ANN CHEM, V640, P145

[8] SIGNIFICANCE OF HISTIDINE IN THYROTROPIN-RELEASING HORMONE (TRH) [J].

GILLESSEN, D ;

PIVA, F ;

STEINER, H ;

STUDER, RO .

HELVETICA CHIMICA ACTA, 1971, 54 (05) :1335-+

[9]

GILLESSEN D, 1970, HELV CHIM ACTA, V54, P236

[10]

Guillemin R, 1971, Vitam Horm, V29, P1

← 1 2 3 →