SYNTHESIS OF (D)-FORMS AND (L)-FORMS OF DIFFERENTIALLY PROTECTED 2-PIPERIDINEMETHANAMINE

被引：21

作者：

PERUMATTAM, J

SHEARER, BG

CONFER, WL

MATHEW, RM

机构：

[1] Nova Pharmaceutical Corporation, 6200 Freeport Centre, Baltimore

来源：

TETRAHEDRON LETTERS | 1991年 / 32卷 / 49期

关键词：

PIPERIDINEMETHANAMINE; PYRROLIDINEMETHANAMINE; PROTEIN KINASE-C INHIBITOR;

D O I：

10.1016/0040-4039(91)80471-H

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

(D)- and (L)-isomers of pipecolic acid were converted into (D)- and (L)-2-piperidinemethanamine using an efficient sequence. The amino groups were selectively protected for further functionalization.

引用

页码：7183 / 7186

页数：4

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