BENZYNE ROUTE TO INDOLES FROM ORTHO-BROMOARYL OR META-BROMOARYL KETONES

被引：23

作者：

FLEMING, I

WOOLIAS, M

机构：

[1] University Chemical Laboratory, Cambridge CB2 1EW, Lensfield Road

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 1979年 / 03期

关键词：

D O I：

10.1039/p19790000827

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Indoles (11) or (14) are formed directly when 2-amino-1-o- (or m-)bromoaryl-ethanols (8) or (13) are treated with potassamide in liquid ammonia.

引用

页码：827 / 828

页数：2

共 11 条

[1]

BLAIKIE KG, 1924, J CHEM SOC, P296

[2] RING CLOSURE VIA ARYNE INTERMEDIATES - A GENERAL PRINCIPLE OF SYNTHESIS [J].

BUNNETT, JF ;

HRUTFIORD, BF .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1961, 83 (07) :1691-&

[3]

Fischer E., 1886, BER, V19, P1563

[4] NEW SYNTHESIS OF INDOLES PARTICULARLY SUITABLE FOR THE SYNTHESIS OF TRYPTAMINES AND TRYPTAMINE ITSELF [J].

FLEMING, I ;

WOOLIAS, M .

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 1979, (03) :829-837

[5] UBER DIE KONSTITUTION DES ARICINS [J].

GOUTAREL, R ;

JANOT, MM ;

LEHIR, A ;

CORRODI, H ;

PRELOG, V .

HELVETICA CHIMICA ACTA, 1954, 37 (06) :1805-1814

[6] NUCLEOPHILE AROMATISCHE SUBSTITUTIONEN .10. KINETIK DER RINGSCHLUSSREAKTIONEN ZU N-METHYL-INDOLIN UND N-METHYL-TETRAHYDROCHINOLIN [J].

HUISGEN, R ;

KONIG, H ;

BLEEKER, N .

CHEMISCHE BERICHTE-RECUEIL, 1959, 92 (02) :424-429

[7] NUCLEOPHILE AROMATISCHE SUBSTITUTIONEN .9. RINGSCHLUSSREAKTIONEN ZU N-METHYL-INDOLIN UND N-METHYL-TETRAHYDROCHINOLIN UND IHR CHEMISMUS [J].

HUISGEN, R ;

KONIG, H .

CHEMISCHE BERICHTE-RECUEIL, 1959, 92 (01) :203-213

[8]

JULIA M, 1966, B SOC CHIM FR, P1335

[9]

KERMACK WO, 1921, J CHEM SOC, P1602

[10]

PAPPALARDO G, 1958, GAZZ CHIM ITAL, V88, P564

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