NON-PEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONISTS .2. PHARMACOLOGY OF S-8308

被引:110
作者
CHIU, AT [1 ]
CARINI, DJ [1 ]
JOHNSON, AL [1 ]
MCCALL, DE [1 ]
PRICE, WA [1 ]
THOOLEN, MJMC [1 ]
WONG, PC [1 ]
TABER, RI [1 ]
TIMMERMANS, PBMWM [1 ]
机构
[1] DUPONT CO, DEPT MED PRODUCTS, DIV PHARM RES, WILMINGTON, DE 19898 USA
关键词
D O I
10.1016/0014-2999(88)90465-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:13 / 21
页数:9
相关论文
共 30 条
  • [1] ANDERSON WP, 1987, KIDNEY INT, V31, pS157
  • [2] BLUMBERG H, 1974, NARCOTIC ANTAGONISTS, V8, P33
  • [3] SPECIFIC-INHIBITION OF RENIN BY AN ANGIOTENSINOGEN ANALOG - STUDIES IN SODIUM DEPLETION AND RENIN-DEPENDENT HYPERTENSION
    BURTON, J
    CODY, RJ
    HERD, JA
    HABER, E
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (09): : 5476 - 5479
  • [4] CANGIANO JL, 1979, J PHARMACOL EXP THER, V208, P310
  • [5] PHARMACOLOGICAL CHARACTERISTICS OF RECEPTOR-OPERATED AND POTENTIAL-OPERATED CA-2+ CHANNELS IN RAT AORTA
    CHIU, AT
    MCCALL, DE
    TIMMERMANS, PBMWM
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 127 (1-2) : 1 - 8
  • [6] DESIGN OF NONPEPTIDAL LIGANDS FOR A PEPTIDE RECEPTOR - CHOLECYSTOKININ ANTAGONISTS
    EVANS, BE
    RITTLE, KE
    BOCK, MG
    DIPARDO, RM
    FREIDINGER, RM
    WHITTER, WL
    GOULD, NP
    LUNDELL, GF
    HOMNICK, CF
    VEBER, DF
    ANDERSON, PS
    CHANG, RSL
    LOTTI, VJ
    CERINO, DJ
    CHEN, TB
    KING, PJ
    KUNKEL, KA
    SPRINGER, JP
    HIRSHFIELD, J
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (07) : 1229 - 1239
  • [7] ISOLATION OF BRADYKININ-POTENTIATING PEPTIDES FROM BOTHROPS-JARARACA VENOM
    FERREIRA, SH
    BARTELT, DC
    GREENE, LJ
    [J]. BIOCHEMISTRY, 1970, 9 (13) : 2583 - &
  • [8] SYNTHESIS AND PHARMACOLOGY OF A NONCOMPETITIVE ANTAGONIST OF ANGIOTENSIN-INDUCED CONTRACTIONS OF VASCULAR SMOOTH-MUSCLE - [SARCOSYL]1-[CYSTEINYL (S-METHYL)]8-ANGIOTENSIN-II
    FREER, RJ
    SUTHERLAND, JC
    DAY, AR
    [J]. CIRCULATION RESEARCH, 1980, 46 (05) : 720 - 725
  • [9] Furakawa Y, 1982, U. S. Patent, Patent No. [4340 598, 4355 040, 4340598]
  • [10] FURUKAWA Y, 1982, Patent No. 4355040