EMPLOYMENT OF A STEROIDAL ALDEHYDE IN A NEW SYNTHESIS OF BETA-LACTAM DERIVATIVES

被引：22

作者：

DOMLING, A ^{[1
]}

KEHAGIA, K ^{[1
]}

UGI, I ^{[1
]}

机构：

[1] TECH UNIV MUNICH, LEHRSTUHL ORGAN CHEM & BIOCHEM 1, D-85747 GARCHING, GERMANY

来源：

TETRAHEDRON | 1995年 / 51卷 / 35期

关键词：

D O I：

10.1016/0040-4020(95)00541-F

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

In this article a beta-lactam-steroid product 4 containing a steroid and a beta-lactam unit is described. Product 4 is easily produced in one step by the means of Ugi reactions. A medium scale high yield procedure for the synthesis of dehydrocholic aldehyde is described.

引用

页码：9519 / 9522

页数：4

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