INTERACTION OF PERMANENTLY UNCHARGED DOPAMINE ANALOGS WITH THE D-2 DOPAMINERGIC RECEPTOR

被引:7
作者
WALLACE, RA
FAROOQUI, T
WALLACE, L
ARES, J
CHANG, YA
MILLER, D
URETSKY, N
机构
[1] OHIO STATE UNIV,COLL PHARM,DIV PHARMACOL,500 W 12TH AVE,COLUMBUS,OH 43210
[2] OHIO STATE UNIV,COLL PHARM,DIV MED CHEM,COLUMBUS,OH 43210
关键词
D O I
10.1016/0006-2952(88)90559-X
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:2077 / 2084
页数:8
相关论文
共 13 条
[1]  
DELEAN A, 1978, AM J PHYSIOL, V235, pE92
[2]   REGIONAL STUDIES OF CATECHOLAMINES IN RAT BRAIN .I. DISPOSITION OF [3H]NOREPINEPHRINE [3H]DOPAMINE AND [3H]DOPA IN VARIOUS REGIONS OF BRAIN [J].
GLOWINSKI, J ;
IVERSEN, LL .
JOURNAL OF NEUROCHEMISTRY, 1966, 13 (08) :655-+
[3]   COMPLETE CONVERSION OF BRAIN D2 DOPAMINE-RECEPTORS FROM THE HIGH-AFFINITY TO THE LOW-AFFINITY STATE FOR DOPAMINE AGONISTS, USING SODIUM-IONS AND GUANINE-NUCLEOTIDE [J].
GRIGORIADIS, D ;
SEEMAN, P .
JOURNAL OF NEUROCHEMISTRY, 1985, 44 (06) :1925-1935
[4]   EFFECT OF CHOLINERGIC DRUGS ON [H-3] ACETYLCHOLINE-RELEASE FROM SLICES OF RAT HIPPOCAMPUS, STRIATUM AND CORTEX [J].
HADHAZY, P ;
SZERB, JC .
BRAIN RESEARCH, 1977, 123 (02) :311-322
[5]   INTERACTIONS OF AGONISTS WITH D-2 DOPAMINE-RECEPTORS - EVIDENCE FOR A SINGLE RECEPTOR POPULATION EXISTING IN MULTIPLE AGONIST AFFINITY-STATES IN RAT STRIATAL MEMBRANES [J].
HAMBLIN, MW ;
LEFF, SE ;
CREESE, I .
BIOCHEMICAL PHARMACOLOGY, 1984, 33 (06) :877-887
[6]   CHRONIC NEUROLEPTIC TREATMENT INCREASES D-2 BUT NOT D-1 RECEPTORS IN RAT STRIATUM [J].
MACKENZIE, RG ;
ZIGMOND, MJ .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 113 (02) :159-165
[7]   LIGAND - A VERSATILE COMPUTERIZED APPROACH FOR CHARACTERIZATION OF LIGAND-BINDING SYSTEMS [J].
MUNSON, PJ ;
RODBARD, D .
ANALYTICAL BIOCHEMISTRY, 1980, 107 (01) :220-239
[8]  
NICHOLS DE, 1983, DOPAMINE RECEPTORS, P201
[9]   SYNTHESIS OF RADIOACTIVE ACETYLCHOLINE FROM [H-3]CHOLINE AND ITS RELEASE FROM CEREBRAL CORTEX SLICES IN-VITRO [J].
RICHTER, JA ;
MARCHBANKS, RM .
JOURNAL OF NEUROCHEMISTRY, 1971, 18 (05) :691-+
[10]   EFFECT OF PERMANENTLY CHARGED AND UNCHARGED DOPAMINERGIC AGONISTS ON THE POTASSIUM-INDUCED RELEASE OF [H-3] ACETYLCHOLINE FROM STRIATAL SLICES [J].
SABOL, B ;
BOLDRY, R ;
FAROOQUI, T ;
CHANG, YA ;
MILLER, D ;
URETSKY, N .
BIOCHEMICAL PHARMACOLOGY, 1987, 36 (10) :1679-1685