PREDICTION OF STEADY-STATE BEHAVIOR OF METABOLITE FROM DOSING OF PARENT DRUG

被引:32
作者
LANE, EA
LEVY, RH
机构
[1] UNIV WASHINGTON,SCH PHARM,DEPT PHARMACEUT SCI,SEATTLE,WA 98195
[2] UNIV WASHINGTON,SCH MED,DEPT NEUROL SURG,SEATTLE,WA 98195
关键词
D O I
10.1002/jps.2600690541
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:610 / 612
页数:3
相关论文
共 7 条
  • [1] PHARMACOLOGICALLY ACTIVE DRUG METABOLITES - THERAPEUTIC AND TOXIC ACTIVITIES, PLASMA AND URINE DATA IN MAN, ACCUMULATION IN RENAL-FAILURE
    DRAYER, DE
    [J]. CLINICAL PHARMACOKINETICS, 1976, 1 (06) : 426 - 443
  • [2] UTILIZATION OF AREA UNDER CURVE TO ELUCIDATE DISPOSITION OF AN EXTENSIVELY BIOTRANSFORMED DRUG
    KAPLAN, SA
    JACK, ML
    COTLER, S
    ALEXANDER, K
    [J]. JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1973, 1 (03): : 201 - 216
  • [3] KINETICS OF BIOTRANSFORMATION OF CLONAZEPAM TO ITS 7-AMINO METABOLITE IN THE MONKEY
    LAI, AA
    MIN, BH
    GARLAND, WA
    LEVY, RH
    [J]. JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1979, 7 (01): : 87 - 95
  • [4] LANE EA, EPILEPSY
  • [5] EXPERIMENTAL ANTICONVULSANT CINROMIDE IN MONKEY MODEL - PRELIMINARY EFFICACY
    LOCKARD, JS
    LEVY, RH
    DUCHARME, LL
    CONGDON, WC
    [J]. EPILEPSIA, 1979, 20 (04) : 339 - 350
  • [6] SEQUENTIAL 1ST-PASS ELIMINATION OF A METABOLITE DERIVED FROM A PRECURSOR
    PANG, KS
    GILLETTE, JR
    [J]. JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1979, 7 (03): : 275 - 290
  • [7] PATEL IH, 1978, J PHARMACOL EXP THER, V206, P607