SYNTHESIS OF [1,2,3]TRIAZOLO[1,5-A][4,1]BENZOXAZEPINE VIA INTRAMOLECULAR AZIDE CYCLOADDITION

被引：15

作者：

GARANTI, L

MOLTENI, G

ZECCHI, G

机构：

[1] Dipartimento di Chimica Organica, Industriale dell'Università, I-20133 Milano

来源：

HETEROCYCLES | 1994年 / 38卷 / 02期

关键词：

D O I：

10.3987/COM-93-6533

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Starting from isatoic anhydride and propargyl alcohols, we developed a synthetic approach to the title compounds, where the key step is an intramolecular cycloaddition of the azido group onto the acetylenic bond.

引用

页码：291 / 296

页数：6

共 10 条

[1] BRUCHE L, 1983, J CHEM RES-S, P202
[2] INTRAMOLECULAR 1,3-DIPOLAR CYCLOADDITIONS OF ARYL AZIDES BEARING ALKENYL, ALKYNYL, AND NITRILE GROUPS
FUSCO, R
GARANTI, L
ZECCHI, G
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1975, 40 (13) : 1906 - 1909
[3] GARANTI L, 1975, SYNTHESIS-STUTTGART, P666
[4] THERMOCHEMICAL BEHAVIOR OF ORTHO-AZIDOCINNAMONITRILES
GARANTI, L
ZECCHI, G
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1980, 45 (23) : 4767 - 4769
[5] GOLSE R, 1948, Ann Chim (Paris), V3, P527
[6] HUISGEN R, 1984, 1 3 DIPOLAR CYCLOADD, V1, pCH1
[7] MOHIUDDIN G, 1986, HETEROCYCLES, V24, P3489
[8] PADWA A, 1990, ADV CYCLOADDITION, V2, P1
[9] PADWA A, 1984, 1 3 DIPOLAR CYCLOADD, V2, pCH12
[10] Schultz A. G., 1988, ADV CYCLOADDITION, V1, P53

← 1 →