THE THERMODYNAMIC ESSENCE OF THE REVERSIBLE INACTIVATION OF NA+/K+-TRANSPORTING ATPASE BY VARIOUS DIGITALIS DERIVATIVES IS RELAXATION OF ENZYME CONFORMATIONAL ENERGY

被引:9
作者
BEER, J
KUNZE, R
HERRMANN, I
PORTIUS, HJ
MIRSALICHOVA, NM
ABUBAKIROV, NK
REPKE, KRH
机构
[1] ACAD SCI GDR,CENT INST MOLEC BIOL,ROBERT ROSSLE STR 10,DDR-1115 BERLIN,GER DEM REP
[2] ACAD SCI UZSSR,INST CHEM PLANT PROD,TASHKENT,UZBEKISTAN,USSR
关键词
D O I
10.1016/0005-2736(88)90256-8
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:335 / 346
页数:12
相关论文
共 49 条
[1]  
AKERA T, 1981, HDB EXPT PHARM, V56, P287
[2]   FUNCTIONAL-GROUP CONTRIBUTIONS TO DRUG RECEPTOR INTERACTIONS [J].
ANDREWS, PR ;
CRAIK, DJ ;
MARTIN, JL .
JOURNAL OF MEDICINAL CHEMISTRY, 1984, 27 (12) :1648-1657
[4]  
CARILLI CT, 1982, J BIOL CHEM, V257, P5601
[5]  
CLARK AF, 1975, J BIOL CHEM, V250, P9355
[6]  
Eftink M., 1980, BIOL MICROCALORIM, P343
[7]  
EIGEN M, 1963, ADV ENZYMOL REL S BI, V25, P1
[8]   OUABAIN-RECEPTOR INTERACTIONS IN (NA++K+)-ATPASE PREPARATIONS FROM DIFFERENT TISSUES AND SPECIES - DETERMINATION OF KINETIC CONSTANTS AND DISSOCIATION-CONSTANTS [J].
ERDMANN, E ;
SCHONER, W .
BIOCHIMICA ET BIOPHYSICA ACTA, 1973, 307 (02) :386-398
[9]  
ERDMANN E, 1981, HDB EXPT PHARM, V56, P337
[10]   The activated complex and the absolute rate of chemical reactions [J].
Eyring, H .
CHEMICAL REVIEWS, 1935, 17 (01) :65-77