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SELECTIVE THYROMIMETICS - CARDIAC-SPARING THYROID-HORMONE ANALOGS CONTAINING 3'-ARYLMETHYL SUBSTITUENTS
被引:38
作者
:
LEESON, PD
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
LEESON, PD
[
1
]
EMMETT, JC
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
EMMETT, JC
[
1
]
SHAH, VP
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SHAH, VP
[
1
]
SHOWELL, GA
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SHOWELL, GA
[
1
]
NOVELLI, R
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
NOVELLI, R
[
1
]
PRAIN, HD
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
PRAIN, HD
[
1
]
BENSON, MG
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
BENSON, MG
[
1
]
ELLIS, D
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
ELLIS, D
[
1
]
PEARCE, NJ
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
PEARCE, NJ
[
1
]
UNDERWOOD, AH
论文数:
0
引用数:
0
h-index:
0
机构:
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
UNDERWOOD, AH
[
1
]
机构
:
[1]
SK&F RES LTD, WELWYN AL6 9AR, HERTS, ENGLAND
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1989年
/ 32卷
/ 02期
关键词
:
D O I
:
10.1021/jm00122a009
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:320 / 336
页数:17
相关论文
共 57 条
[1]
BINDING OF THYROID-HORMONES AND ANALOGS TO THE HUMAN-PLASMA PROTEIN PRE-ALBUMIN
ANDREA, TA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
ANDREA, TA
CAVALIERI, RR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
CAVALIERI, RR
GOLDFINE, ID
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
GOLDFINE, ID
JORGENSEN, EC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
JORGENSEN, EC
[J].
BIOCHEMISTRY,
1980,
19
(01)
: 55
-
63
[2]
LIPID AND LIPOPROTEIN PATTERN IN THYROID-DYSFUNCTION AND THE EFFECT OF THERAPY
AVIRAM, M
论文数:
0
引用数:
0
h-index:
0
机构:
RAMBAM MED CTR, INST ENDOCRINOL, HAIFA, ISRAEL
AVIRAM, M
LUBOSHITZKY, R
论文数:
0
引用数:
0
h-index:
0
机构:
RAMBAM MED CTR, INST ENDOCRINOL, HAIFA, ISRAEL
LUBOSHITZKY, R
BROOK, JG
论文数:
0
引用数:
0
h-index:
0
机构:
RAMBAM MED CTR, INST ENDOCRINOL, HAIFA, ISRAEL
BROOK, JG
[J].
CLINICAL BIOCHEMISTRY,
1982,
15
(01)
: 62
-
66
[3]
BANDER A, 1963, ARZNEIMITTELFORSCH, V13, P1
[4]
BECKMANN R, 1979, ARZNEIMITTEL-FORSCH, V29-1, P499
[5]
3'-ACETYL-3,5-DIIODO-L-THYRONINE - A NOVEL HIGHLY-ACTIVE THYROMIMETIC WITH LOW RECEPTOR AFFINITY
BENSON, MG
论文数:
0
引用数:
0
h-index:
0
BENSON, MG
ELLIS, D
论文数:
0
引用数:
0
h-index:
0
ELLIS, D
EMMETT, JC
论文数:
0
引用数:
0
h-index:
0
EMMETT, JC
LEESON, PD
论文数:
0
引用数:
0
h-index:
0
LEESON, PD
PEARCE, NJ
论文数:
0
引用数:
0
h-index:
0
PEARCE, NJ
SHAH, VP
论文数:
0
引用数:
0
h-index:
0
SHAH, VP
UNDERWOOD, AH
论文数:
0
引用数:
0
h-index:
0
UNDERWOOD, AH
[J].
BIOCHEMICAL PHARMACOLOGY,
1984,
33
(20)
: 3143
-
3149
[6]
THYROMIMETICS .V. SYNTHESIS AND BIOLOGICAL SCREENING OF ALPHA-METHYLTHYROXINE
BLANK, B
论文数:
0
引用数:
0
h-index:
0
BLANK, B
RICE, EG
论文数:
0
引用数:
0
h-index:
0
RICE, EG
PFEIFFER, FR
论文数:
0
引用数:
0
h-index:
0
PFEIFFER, FR
GREENBERG, CM
论文数:
0
引用数:
0
h-index:
0
GREENBERG, CM
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1966,
9
(01)
: 10
-
+
[7]
THYROMIMETICS .3. SYNTHESIS + RELATIVE THYROMIMETIC ACTIVITIES OF SOME 4-ETHERS OF IODINATED THYRONINES + THYROALKANOIC ACIDS
BLANK, B
论文数:
0
引用数:
0
h-index:
0
BLANK, B
KERWIN, JF
论文数:
0
引用数:
0
h-index:
0
KERWIN, JF
GREENBERG, CM
论文数:
0
引用数:
0
h-index:
0
GREENBERG, CM
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1964,
7
(01)
: 53
-
&
[8]
THYROMIMETICS .6. SYNTHESIS AND BIOLOGICAL SCREENING OF 3,5-DIIODOTHYROACETIC AND -PROPIONIC ACID ANALOGS
BLANK, B
论文数:
0
引用数:
0
h-index:
0
BLANK, B
PFEIFFER, FR
论文数:
0
引用数:
0
h-index:
0
PFEIFFER, FR
GREENBER.CM
论文数:
0
引用数:
0
h-index:
0
GREENBER.CM
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1966,
9
(06)
: 832
-
&
[9]
BOLGER MB, 1980, J BIOL CHEM, V255, P271
[10]
VARIOUS EFFECTS OF THYROXINE ANALOGUES ON THE HEART AND SERUM CHOLESTEROL IN THE RAT
BOYD, GS
论文数:
0
引用数:
0
h-index:
0
BOYD, GS
OLIVER, MF
论文数:
0
引用数:
0
h-index:
0
OLIVER, MF
[J].
JOURNAL OF ENDOCRINOLOGY,
1960,
21
(01)
: 25
-
32
←
1
2
3
4
5
6
→
共 57 条
[1]
BINDING OF THYROID-HORMONES AND ANALOGS TO THE HUMAN-PLASMA PROTEIN PRE-ALBUMIN
ANDREA, TA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
ANDREA, TA
CAVALIERI, RR
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
CAVALIERI, RR
GOLDFINE, ID
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
GOLDFINE, ID
JORGENSEN, EC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV CALIF SAN FRANCISCO,SCH PHARM,DEPT PHARMACEUT CHEM,SAN FRANCISCO,CA 94143
JORGENSEN, EC
[J].
BIOCHEMISTRY,
1980,
19
(01)
: 55
-
63
[2]
LIPID AND LIPOPROTEIN PATTERN IN THYROID-DYSFUNCTION AND THE EFFECT OF THERAPY
AVIRAM, M
论文数:
0
引用数:
0
h-index:
0
机构:
RAMBAM MED CTR, INST ENDOCRINOL, HAIFA, ISRAEL
AVIRAM, M
LUBOSHITZKY, R
论文数:
0
引用数:
0
h-index:
0
机构:
RAMBAM MED CTR, INST ENDOCRINOL, HAIFA, ISRAEL
LUBOSHITZKY, R
BROOK, JG
论文数:
0
引用数:
0
h-index:
0
机构:
RAMBAM MED CTR, INST ENDOCRINOL, HAIFA, ISRAEL
BROOK, JG
[J].
CLINICAL BIOCHEMISTRY,
1982,
15
(01)
: 62
-
66
[3]
BANDER A, 1963, ARZNEIMITTELFORSCH, V13, P1
[4]
BECKMANN R, 1979, ARZNEIMITTEL-FORSCH, V29-1, P499
[5]
3'-ACETYL-3,5-DIIODO-L-THYRONINE - A NOVEL HIGHLY-ACTIVE THYROMIMETIC WITH LOW RECEPTOR AFFINITY
BENSON, MG
论文数:
0
引用数:
0
h-index:
0
BENSON, MG
ELLIS, D
论文数:
0
引用数:
0
h-index:
0
ELLIS, D
EMMETT, JC
论文数:
0
引用数:
0
h-index:
0
EMMETT, JC
LEESON, PD
论文数:
0
引用数:
0
h-index:
0
LEESON, PD
PEARCE, NJ
论文数:
0
引用数:
0
h-index:
0
PEARCE, NJ
SHAH, VP
论文数:
0
引用数:
0
h-index:
0
SHAH, VP
UNDERWOOD, AH
论文数:
0
引用数:
0
h-index:
0
UNDERWOOD, AH
[J].
BIOCHEMICAL PHARMACOLOGY,
1984,
33
(20)
: 3143
-
3149
[6]
THYROMIMETICS .V. SYNTHESIS AND BIOLOGICAL SCREENING OF ALPHA-METHYLTHYROXINE
BLANK, B
论文数:
0
引用数:
0
h-index:
0
BLANK, B
RICE, EG
论文数:
0
引用数:
0
h-index:
0
RICE, EG
PFEIFFER, FR
论文数:
0
引用数:
0
h-index:
0
PFEIFFER, FR
GREENBERG, CM
论文数:
0
引用数:
0
h-index:
0
GREENBERG, CM
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1966,
9
(01)
: 10
-
+
[7]
THYROMIMETICS .3. SYNTHESIS + RELATIVE THYROMIMETIC ACTIVITIES OF SOME 4-ETHERS OF IODINATED THYRONINES + THYROALKANOIC ACIDS
BLANK, B
论文数:
0
引用数:
0
h-index:
0
BLANK, B
KERWIN, JF
论文数:
0
引用数:
0
h-index:
0
KERWIN, JF
GREENBERG, CM
论文数:
0
引用数:
0
h-index:
0
GREENBERG, CM
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1964,
7
(01)
: 53
-
&
[8]
THYROMIMETICS .6. SYNTHESIS AND BIOLOGICAL SCREENING OF 3,5-DIIODOTHYROACETIC AND -PROPIONIC ACID ANALOGS
BLANK, B
论文数:
0
引用数:
0
h-index:
0
BLANK, B
PFEIFFER, FR
论文数:
0
引用数:
0
h-index:
0
PFEIFFER, FR
GREENBER.CM
论文数:
0
引用数:
0
h-index:
0
GREENBER.CM
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1966,
9
(06)
: 832
-
&
[9]
BOLGER MB, 1980, J BIOL CHEM, V255, P271
[10]
VARIOUS EFFECTS OF THYROXINE ANALOGUES ON THE HEART AND SERUM CHOLESTEROL IN THE RAT
BOYD, GS
论文数:
0
引用数:
0
h-index:
0
BOYD, GS
OLIVER, MF
论文数:
0
引用数:
0
h-index:
0
OLIVER, MF
[J].
JOURNAL OF ENDOCRINOLOGY,
1960,
21
(01)
: 25
-
32
←
1
2
3
4
5
6
→