HA-966 ACTS AT A MODULATORY GLYCINE SITE TO INHIBIT N-METHYL-D-ASPARTATE-EVOKED NEUROTRANSMITTER RELEASE

被引:44
作者
KEITH, RA
MANGANO, TJ
MEINERS, BA
STUMPO, RJ
KLIKA, AB
PATEL, J
SALAMA, AI
机构
关键词
D O I
10.1016/0014-2999(89)90351-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:393 / 400
页数:8
相关论文
共 30 条
[1]  
BERTOLINO M, 1988, MOL PHARMACOL, V34, P98
[2]   BIOCHEMICAL-EVIDENCE THAT GLYCINE ALLOSTERICALLY REGULATES AN NMDA RECEPTOR-COUPLED ION CHANNEL [J].
BONHAUS, DW ;
BURGE, BC ;
MCNAMARA, JO .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 142 (03) :489-490
[3]   LIGHT MICROSCOPIC AUTORADIOGRAPHIC LOCALIZATION OF [H-3] GLYCINE AND [H-3] STRYCHNINE BINDING-SITES IN RAT-BRAIN [J].
BRISTOW, DR ;
BOWERY, NG ;
WOODRUFF, GN .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1986, 126 (03) :303-307
[4]   CPP, A NEW POTENT AND SELECTIVE NMDA ANTAGONIST - DEPRESSION OF CENTRAL NEURON RESPONSES, AFFINITY FOR [H-3] D-AP5 BINDING-SITES ON BRAIN MEMBRANES AND ANTICONVULSANT ACTIVITY [J].
DAVIES, J ;
EVANS, RH ;
HERRLING, PL ;
JONES, AW ;
OLVERMAN, HJ ;
POOK, P ;
WATKINS, JC .
BRAIN RESEARCH, 1986, 382 (01) :169-173
[6]   FREE AND CONJUGATED AMINO-ACIDS IN HUMAN CSF - INFLUENCE OF AGE AND SEX [J].
FERRARO, TN ;
HARE, TA .
BRAIN RESEARCH, 1985, 338 (01) :53-60
[7]   GLYCINE REVERSES ANTAGONISM OF N-METHYL-D-ASPARTATE (NMDA) BY 1-HYDROXY-3-AMINOPYRROLIDONE-2 (HA-966) BUT NOT BY D-2-AMINO-5-PHOPHONOVALERATE (D-AP5) ON RAT CORTICAL SLICES [J].
FLETCHER, EJ ;
LODGE, D .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 151 (01) :161-162
[8]   GLYCINE POTENTIATES THE NMDA RESPONSE IN CULTURED MOUSE-BRAIN NEURONS [J].
JOHNSON, JW ;
ASCHER, P .
NATURE, 1987, 325 (6104) :529-531
[9]  
JONES SM, 1987, J PHARMACOL EXP THER, V240, P492
[10]  
KEITH RA, 1988, NEUR ABSTR, V14, P792