PHARMACOLOGICAL PROFILE OF THE SUBSTITUTED BETA-LACTAM L-659,286 - A MEMBER OF A NEW CLASS OF HUMAN-PMN ELASTASE INHIBITORS

被引：42

作者：

BONNEY, RJ ^{[1
]}

ASHE, B ^{[1
]}

MAYCOCK, A ^{[1
]}

DELLEA, P ^{[1
]}

HAND, K ^{[1
]}

OSINGA, D ^{[1
]}

FLETCHER, D ^{[1
]}

MUMFORD, R ^{[1
]}

DAVIES, P ^{[1
]}

FRANKENFIELD, D ^{[1
]}

NOLAN, T ^{[1
]}

SCHAEFFER, L ^{[1
]}

HAGMANN, W ^{[1
]}

FINKE, P ^{[1
]}

SHAH, S ^{[1
]}

DORN, C ^{[1
]}

DOHERTY, J ^{[1
]}

机构：

[1] MERCK SHARP & DOHME RES LABS,W POINT,PA 19486

来源：

JOURNAL OF CELLULAR BIOCHEMISTRY | 1989年 / 39卷 / 01期

关键词：

D O I：

10.1002/jcb.240390106

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：47 / 53

页数：7

共 8 条

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[7]

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[8] MECHANISM OF INACTIVATION OF HUMAN-LEUKOCYTE ELASTASE BY A CHLOROMETHYL KETONE - KINETIC AND SOLVENT ISOTOPE EFFECT STUDIES [J].

STEIN, RL ;

TRAINOR, DA .

BIOCHEMISTRY, 1986, 25 (19) :5414-5419

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