EFFECTS OF N-ARALKYL SUBSTITUTION OF BETA-AGONISTS ON ALPHA-ADRENOCEPTOR AND BETA-ADRENOCEPTOR SUBTYPES - PHARMACOLOGICAL STUDIES AND BINDING ASSAYS

被引:48
作者
DECKER, N [1 ]
QUENNEDEY, MC [1 ]
ROUOT, B [1 ]
SCHWARTZ, J [1 ]
VELLY, J [1 ]
机构
[1] FAC MED STRASBOURG, INST PHARMACOL,INSERM,U206,CNRS,ERA 142, 11 RUE HUMANN, F-67000 STRASBOURG, FRANCE
关键词
D O I
10.1111/j.2042-7158.1982.tb04195.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:107 / 112
页数:6
相关论文
共 31 条
[1]   N-ARALKYL SUBSTITUTION INCREASES THE AFFINITY OF ADRENERGIC-DRUGS FOR THE ALPHA-ADRENOCEPTOR IN RAT-LIVER [J].
AGGERBECK, M ;
GUELLAEN, G ;
HANOUNE, J .
BRITISH JOURNAL OF PHARMACOLOGY, 1979, 65 (01) :155-159
[3]  
ARIENS EJ, 1957, ARCH INT PHARMACOD T, V110, P275
[4]   SOME QUANTITATIVE USES OF DRUG ANTAGONISTS [J].
ARUNLAKSHANA, O ;
SCHILD, HO .
BRITISH JOURNAL OF PHARMACOLOGY AND CHEMOTHERAPY, 1959, 14 (01) :48-58
[5]   FUNCTIONAL BASIS FOR CLASSIFICATION OF ALPHA-ADRENERGIC RECEPTORS [J].
BERTHELSEN, S ;
PETTINGER, WA .
LIFE SCIENCES, 1977, 21 (05) :595-606
[6]   EFFECTS OF LABETALOL (AH5158) ON ADRENERGIC TRANSMISSION IN CAT SPLEEN [J].
BLAKELEY, AGH ;
SUMMERS, RJ .
BRITISH JOURNAL OF PHARMACOLOGY, 1977, 59 (04) :643-650
[7]  
BRITTAIN RT, 1976, BRIT J CLIN PHARMACO, V3, P681
[8]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[9]   CARDIOVASCULAR PROPERTIES OF MEDROXALOL, A NEW ANTIHYPERTENSIVE DRUG [J].
DAGE, RC ;
CHENG, HC ;
WOODWARD, JK .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1981, 3 (02) :299-315
[10]   HUMAN-PLATELET ALPHA-2-ADRENERGIC RECEPTORS - LABELING WITH YOHIMBINE-H-3, A SELECTIVE ANTAGONIST LIGAND [J].
DAIGUJI, M ;
MELTZER, HY ;
UPRICHARD, DC .
LIFE SCIENCES, 1981, 28 (24) :2705-2717