DIFFERENT EFFECTS OF INTRACEREBRAL AND SYSTEMIC ADMINISTRATION OF BUSPIRONE IN THE FORCED SWIMMING TEST - INVOLVEMENT OF A METABOLITE

被引:55
作者
CERVO, L
GRIGNASCHI, G
SAMANIN, R
机构
关键词
D O I
10.1016/0024-3205(88)90359-1
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2095 / 2102
页数:8
相关论文
共 22 条
[1]   BLOCKADE OF ALPHA-2-ADRENOCEPTORS BY 1-(2-PYRIMIDINYL)-PIPERAZINE (PMP) INVIVO AND ITS RELATION TO THE ACTIVITY OF BUSPIRONE [J].
BIANCHI, G ;
GARATTINI, S .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 147 (03) :343-350
[2]   EVIDENCE OF DOPAMINE INVOLVEMENT IN THE EFFECT OF REPEATED TREATMENT WITH VARIOUS ANTIDEPRESSANTS IN THE BEHAVIORAL DESPAIR TEST IN RATS [J].
BORSINI, F ;
PULVIRENTI, L ;
SAMANIN, R .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 110 (02) :253-256
[3]   1-(2-PYRIMIDINYL)-PIPERAZINE AS ACTIVE METABOLITE OF BUSPIRONE IN MAN AND RAT [J].
CACCIA, S ;
CONTI, I ;
VIGANO, G ;
GARATTINI, S .
PHARMACOLOGY, 1986, 33 (01) :46-51
[4]   DISPOSITION AND METABOLISM OF BUSPIRONE AND ITS METABOLITE 1-(2-PYRIMIDINYL)-PIPERAZINE IN THE RAT [J].
CACCIA, S ;
MUGLIA, M ;
MANCINELLI, A ;
GARATTINI, S .
XENOBIOTICA, 1983, 13 (03) :147-153
[5]   POTENTIAL ANTIDEPRESSANT PROPERTIES OF 8-HYDROXY-2-(DI-N-PROPYLAMINO)TETRALIN, A SELECTIVE SEROTONIN-1A RECEPTOR AGONIST [J].
CERVO, L ;
SAMANIN, R .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1987, 144 (02) :223-229
[6]   NEURO-PHARMACOLOGICAL STUDIES IN RODENTS ON THE ACTION OF RX-781094, A NEW SELECTIVE ALPHA-2 ADRENOCEPTOR ANTAGONIST [J].
DETTMAR, PW ;
LYNN, AG ;
TULLOCH, IF .
NEUROPHARMACOLOGY, 1983, 22 (06) :729-737
[7]   2-ALKYL ANALOGS OF IDAZOXAN (RX-781094) WITH ENHANCED ANTAGONIST POTENCY AND SELECTIVITY AT CENTRAL ALPHA-2-ADRENOCEPTORS IN THE RAT [J].
GADIE, B ;
LANE, AC ;
MCCARTHY, PS ;
TULLOCH, IF ;
WALTER, DS .
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 83 (03) :707-712
[8]   [H-3]8-HYDROXY-2-(DI-NORMAL-PROPYLAMINO)TETRALIN BINDING TO PRESYNAPTIC AND POSTSYNAPTIC 5-HYDROXYTRYPTAMINE SITES IN VARIOUS REGIONS OF THE RAT-BRAIN [J].
HALL, MD ;
ELMESTIKAWY, S ;
EMERIT, MB ;
PICHAT, L ;
HAMON, M ;
GOZLAN, H .
JOURNAL OF NEUROCHEMISTRY, 1985, 44 (06) :1685-1696
[9]   EFFECTS OF ALPHA-ADRENOCEPTOR AGONISTS AND ANTAGONISTS IN A MAZE-EXPLORATION MODEL OF FEAR-MOTIVATED BEHAVIOR [J].
HANDLEY, SL ;
MITHANI, S .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1984, 327 (01) :1-5
[10]  
Konig JFR, 1963, RAT BRAIN STEREOTAXI