HIGH-AFFINITY BINDING TO THE ESTROGEN-RECEPTOR OF [4-HYDROXYTAMOXIFEN-H-3, AN ACTIVE ANTI-ESTROGEN METABOLITE

被引:122
作者
BORGNA, JL
ROCHEFORT, H
机构
关键词
D O I
10.1016/0303-7207(80)90095-7
中图分类号
Q2 [细胞生物学];
学科分类号
071009 ; 090102 ;
摘要
引用
收藏
页码:71 / 85
页数:15
相关论文
共 33 条
[1]  
Alberts B., 1971, METHOD ENZYMOL, V21, P198
[2]   INVITRO BINDING OF ESTROGEN-RECEPTOR TO DNA - ABSENCE OF SATURATION AT EQUILIBRIUM [J].
ANDRE, J ;
ROCHEFORT, H .
FEBS LETTERS, 1975, 50 (03) :319-323
[3]   MONOHYDROXYTAMOXIFEN - ANTIOESTROGEN WITH HIGH-AFFINITY FOR THE CHICK OVIDUCT ESTROGEN-RECEPTOR [J].
BINART, N ;
CATELLI, MG ;
GEYNET, C ;
PURI, V ;
HAHNEL, R ;
MESTER, J ;
BAULIEU, EE .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1979, 91 (03) :812-818
[4]   DETERMINATION OF PROTEIN-LIGAND BINDING CONSTANTS AT EQUILIBRIUM IN BIOLOGICAL SAMPLES [J].
BLONDEAU, JP ;
ROBEL, P .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1975, 55 (02) :375-384
[5]  
BORGNA JL, 1979, CR HEBD ACAD SCI, V287, P1141
[6]  
BORGNA JL, UNPUBLISHED
[7]   RELEVANCE OF KINETIC-PARAMETERS IN DETERMINATION OF SPECIFIC BINDING TO ESTROGEN-RECEPTOR [J].
BOUTON, MM ;
RAYNAUD, JP .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1978, 9 (01) :9-15
[8]   ANDROGENIC, ANTI-ANDROGENIC, AND SYNANDROGENIC ACTIONS OF PROGESTINS - ROLE OF STERIC AND ALLOSTERIC INTERACTIONS WITH ANDROGEN RECEPTORS [J].
BULLOCK, LP ;
BARDIN, CW ;
SHERMAN, MR .
ENDOCRINOLOGY, 1978, 103 (05) :1768-1782
[9]   HIGH-AFFINITY BINDING OF ANTI-ESTROGEN [TAMOXIFEN-H-3 TO 8S ESTRADIOL RECEPTOR [J].
CAPONY, F ;
ROCHEFORT, H .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1978, 11 (02) :181-198
[10]   INVIVO EFFECT OF ANTI-ESTROGENS ON LOCALIZATION AND REPLENISHMENT OF ESTROGEN-RECEPTOR [J].
CAPONY, F ;
ROCHEFORT, H .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1975, 3 (03) :233-251