CHARACTERIZATION OF THE ENANTIOMERIC 3-SUBSTITUTED-1,4-BENZODIAZEPIN-2-ONES BINDING TO THE GABA BDZ CHLORIDE IONOPHORE RECEPTOR COMPLEX

被引：4

作者：

BERTUCCI, C

SALVADORI, P

BELFIORE, S

MARTINI, C

LUCACCHINI, A

机构：

[1] CNR, CTR STUDIO MACROMOLEC STEREORDINATE OTTICAMENTE AT, DIPARTIMENTO CHIM & CHIM IND, I-56126 PISA, ITALY

[2] IST POLICATTEDRA DISCIPLINE BIOL, I-56126 PISA, ITALY

来源：

JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS | 1992年 / 10卷 / 05期

关键词：

CHIRAL BENZODIAZEPINES; STEREOCHEMISTRY; GABA BENZODIAZEPINE CHLORIDE IONOPHORE RECEPTOR COMPLEX; CHIRAL CHROMATOGRAPHY; ENANTIOSELECTIVE RECEPTOR BINDING; INVITRO RECEPTOR FUNCTION;

D O I：

10.1016/0731-7085(92)80053-P

中图分类号：

O65 [分析化学];

学科分类号：

070302 ; 081704 ;

摘要：

[No abstract available]

引用

页码：359 / 363

页数：5

共 33 条

[1]

BLASCHKE G, 1986, ARZNEIMITTEL-FORSCH, V36-1, P893

[2]

BLOUNT JF, 1983, MOL PHARMACOL, V24, P425

[3] BENZODIAZEPINE RECEPTOR LIGANDS WITH POSITIVE AND NEGATIVE EFFICACY [J].

BRAESTRUP, C ;

NIELSEN, M ;

HONORE, T ;

JENSEN, LH ;

PETERSEN, EN .

NEUROPHARMACOLOGY, 1983, 22 (12B) :1451-1457

[4] INTERACTION OF CONVULSIVE LIGANDS WITH BENZODIAZEPINE RECEPTORS [J].

BRAESTRUP, C ;

SCHMIECHEN, R ;

NEEF, G ;

NIELSEN, M ;

PETERSEN, EN .

SCIENCE, 1982, 216 (4551) :1241-1243

[5]

BRAESTRUP C, 1983, HDB PSYCHOPHARMACOLO, P258

[6]

CAHAN RS, 1966, ANGEW CHEM, V78, P413

[7]

CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099

[8] GAMMA-AMINOBUTYRIC ACID REGULATION OF THE BENZODIAZEPINE RECEPTOR - BIOCHEMICAL-EVIDENCE FOR PHARMACOLOGICALLY DIFFERENT EFFECTS OF BENZODIAZEPINES AND PROPYL BETA-CARBOLINE-3-CARBOXYLATE [J].

EHLERT, FJ ;

ROESKE, WR ;

BRAESTRUP, C ;

YAMAMURA, SH ;

YAMAMURA, HI .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 70 (04) :593-595

[9]

GEE KW, 1986, MOL PHARMACOL, V30, P218

[10] ATROPISOMERS OF 1,4-BENZODIAZEPINES - SYNTHESIS AND RESOLUTION OF A DIAZEPAM-RELATED 1,4-BENZODIAZEPINE [J].

GILMAN, NW ;

ROSEN, P ;

EARLEY, JV ;

COOK, C ;

TODARO, LJ .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1990, 112 (10) :3969-3978

← 1 2 3 4 →