METABOLISM OF THE CONTRACEPTIVE STEROID DESOGESTREL BY THE INTESTINAL-MUCOSA

被引:26
作者
MADDEN, S
BACK, DJ
MARTIN, CA
ORME, MLE
机构
基金
英国惠康基金;
关键词
D O I
10.1111/j.1365-2125.1989.tb05368.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:295 / 299
页数:5
相关论文
共 11 条
[1]  
BACK D J, 1987, Alimentary Pharmacology and Therapeutics, V1, P339
[2]   THE GUT WALL METABOLISM OF ETHINYLESTRADIOL AND ITS CONTRIBUTION TO THE PRE-SYSTEMIC METABOLISM OF ETHINYLESTRADIOL IN HUMANS [J].
BACK, DJ ;
BRECKENRIDGE, AM ;
MACIVER, M ;
ORME, M ;
PURBA, HS ;
ROWE, PH ;
TAYLOR, I .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1982, 13 (03) :325-330
[3]   PLASMA-CONCENTRATIONS OF 3-KETO-DESOGESTREL AFTER ORAL-ADMINISTRATION OF DESOGESTREL AND INTRAVENOUS ADMINISTRATION OF 3-KETO-DESOGESTREL [J].
BACK, DJ ;
GRIMMER, SFM ;
SHENOY, N ;
ORME, MLE .
CONTRACEPTION, 1987, 35 (06) :619-626
[4]  
GRADY GF, 1970, GASTROENTEROLOGY, V59, P583
[5]  
HARTMANN F, 1983, DRUG METAB DISPOS, V11, P244
[6]   SERUM LEVELS OF 3-KETO-DESOGESTREL AFTER ORAL-ADMINISTRATION OF DESOGESTREL AND 3-KETO-DESOGESTREL [J].
HASENACK, HG ;
BOSCH, AMG ;
KAAR, K .
CONTRACEPTION, 1986, 33 (06) :591-596
[7]   SULFATION AND GLUCURONIDATION OF ETHINYLESTRADIOL IN HUMAN-LIVER INVITRO [J].
PACIFICI, GM ;
BACK, DJ .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1988, 31 (03) :345-349
[8]   INTESTINAL METABOLISM OF ETHINYLESTRADIOL AND PARACETAMOL INVITRO - STUDIES USING USSING CHAMBERS [J].
ROGERS, SM ;
BACK, DJ ;
ORME, ML .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1987, 23 (06) :727-734
[9]   ACTIVE TRANSPORT OF SODIUM AS THE SOURCE OF ELECTRIC CURRENT IN THE SHORT-CIRCUITED ISOLATED FROG SKIN [J].
USSING, HH ;
ZERAHN, K .
ACTA PHYSIOLOGICA SCANDINAVICA, 1951, 23 (2-3) :110-127
[10]   BIOLOGICAL EFFECTS OF A NEW AND POTENT PROGESTAGEN - CLINICAL-STUDY [J].
VIINIKKA, L ;
YLIKORKALA, O ;
NUMMI, S ;
VIRKKUNEN, P ;
RANTA, T ;
ALAPIESSA, U ;
VIHKO, R .
ACTA ENDOCRINOLOGICA, 1976, 83 (02) :429-438