SYNTHESIS OF 2H-3,4-DIHYDRO-1,2-BENZOSELENAZIN-3-ONE AND DERIVATIVES - A NEW HETEROCYCLIC RING-SYSTEM

被引：78

作者：

JACQUEMIN, PV

CHRISTIAENS, LE

RENSON, MJ

EVERS, MJ

DEREU, N

机构：

[1] UNIV LIEGE,INST ORGAN CHEM B6,SART TILMAN,B-4000 LIEGE,BELGIUM

[2] RHONE POULENC RORER,CTR RECH VITRY ALFORTVILLE,F-94403 VITRY,FRANCE

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 27期

关键词：

BENZOSELENAZINONE; ORGANOSELENIUM; HOMOEBSELEN; SELENOHETEROCYCLE;

D O I：

10.1016/S0040-4039(00)74805-2

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of 2H-3,4-dihydro-1,2-benzoselenazin-3-ones which are six-membered homologues of Ebselen is described in order to evaluate their glutathione peroxidase-like activity. Spectral data of these new heterocycles are given.

引用

页码：3863 / 3866

页数：4

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