HYPERVALENT IODINE OXIDATION OF 2-ARYL-1,2,3,4-TETRA-HYDRO-4-QUINOLONES - AN EASY ACCESS TO 2-ARYL-4-QUINOLONES

被引：44

作者：

PRAKASH, O

KUMAR, D

SAINI, RK

SINGH, SP

机构：

[1] Department of Chemistry, Kurukshetra University

来源：

SYNTHETIC COMMUNICATIONS | 1994年 / 24卷 / 15期

关键词：

D O I：

10.1080/00397919408010231

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Oxidation of 2-aryl-1,2,3,4-tetrahydro-4-quinolones (1a-e) using iodobenzene diacetate in methanolic potassium hydroxide leads to dehydrogenation of 1 thereby providing an easy access to 2-aryl-4-quinolones (2a-e).

引用

页码：2167 / 2172

页数：6

共 13 条

[1] CHALCONE DERIVATIVES AS PRECURSORS OF 1,2,3,4-TETRAHYDRO-4-QUINOLONES [J].

DONNELLY, JA ;

FARRELL, DF .

TETRAHEDRON, 1990, 46 (03) :885-894

[2] THE CHEMISTRY OF 2'-AMINO ANALOGS OF 2'-HYDROXYCHALCONE AND ITS DERIVATIVES [J].

DONNELLY, JA ;

FARRELL, DF .

JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (06) :1757-1761

[3] 2-ARYL-4-QUINOLONES AND FUSED QUINOLINES FROM BETA-CHLOROARYLIDENEMALONATES AND RELATED CHLORO ESTERS [J].

HORMI, OEO ;

PELTONEN, C ;

HEIKKILA, L .

JOURNAL OF ORGANIC CHEMISTRY, 1990, 55 (08) :2513-2515

[4]

KALNIN VN, 1992, TETRAHEDRON LETT, V33, P373

[5]

KASAHARA A, 1981, CHEM IND-LONDON, P121

[6] ALPHA-HYDROXYDIMETHYLACETAL FORMATION FROM AMINOKETONES USING HYPERVALENT IODINE [J].

MORIARTY, RM ;

PRAKASH, O ;

KARALIS, P ;

PRAKASH, I .

TETRAHEDRON LETTERS, 1984, 25 (42) :4745-4748

[7] HYPERVALENT IODINE OXIDATION OF FLAVANONE - SYNTHESIS OF CIS-3-HYDROXYFLAVANONES AND TRANS-3-HYDROXYFLAVANONES [J].

MORIARTY, RM ;

PRAKASH, O .

JOURNAL OF ORGANIC CHEMISTRY, 1985, 50 (02) :151-153

[8] HYPERVALENT IODINE IN ORGANIC-SYNTHESIS [J].

MORIARTY, RM ;

PRAKASH, O .

ACCOUNTS OF CHEMICAL RESEARCH, 1986, 19 (08) :244-250

[9]

PRAKASH O, 1991, INDIAN J CHEM B, V30, P1023

[10] A NEW ROUTE TO 2-ARYL-4-QUINOLONES VIA THALLIUM(III) P-TOLYSULPHONATE MEDIATED OXIDATION OF 2-ARYL-1,2,3,4-TETRAHYDRO-4-QUINOLONES [J].

SINGH, OV ;

KAPIL, RS .

SYNTHETIC COMMUNICATIONS, 1993, 23 (03) :277-283

← 1 2 →