AMILORIDE AND ITS ANALOGS AS TOOLS TO INHIBIT NA+ TRANSPORT VIA THE NA+ CHANNEL, THE NA+/H+ ANTIPORT AND THE NA+/CA-2+ EXCHANGER

被引:96
作者
FRELIN, C [1 ]
BARBRY, P [1 ]
VIGNE, P [1 ]
CHASSANDE, O [1 ]
CRAGOE, EJ [1 ]
LAZDUNSKI, M [1 ]
机构
[1] MERCK SHARP & DOHME RES LABS,W POINT,PA 19486
关键词
D O I
10.1016/0300-9084(88)90196-4
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:1285 / 1290
页数:6
相关论文
共 31 条
[1]   UPTAKE OF [BENZAMIL-H-3 AT DIFFERENT SODIUM CONCENTRATION - INFERENCES REGARDING THE REGULATION OF SODIUM PERMEABILITY [J].
ACEVES, J ;
CUTHBERT, AW .
JOURNAL OF PHYSIOLOGY-LONDON, 1979, 295 (OCT) :491-504
[2]   KINETIC-PROPERTIES OF THE PLASMA-MEMBRANE NA+-H+ EXCHANGER [J].
ARONSON, PS .
ANNUAL REVIEW OF PHYSIOLOGY, 1985, 47 :545-560
[3]   [H-3] PHENAMIL, A RADIOLABELED DIURETIC FOR THE ANALYSIS OF THE AMILORIDE-SENSITIVE NA+ CHANNELS IN KIDNEY MEMBRANES [J].
BARBRY, P ;
FRELIN, C ;
VIGNE, P ;
CRAGOE, EJ ;
LAZDUNSKI, M .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1986, 135 (01) :25-32
[4]   PURIFICATION AND SUBUNIT STRUCTURE OF THE [H-3] PHENAMIL RECEPTOR ASSOCIATED WITH THE RENAL APICAL NA+ CHANNEL [J].
BARBRY, P ;
CHASSANDE, O ;
VIGNE, P ;
FRELIN, C ;
ELLORY, C ;
CRAGOE, EJ ;
LAZDUNSKI, M .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1987, 84 (14) :4836-4840
[5]   AMILORIDE - A MOLECULAR PROBE OF SODIUM-TRANSPORT IN TISSUES AND CELLS [J].
BENOS, DJ .
AMERICAN JOURNAL OF PHYSIOLOGY, 1982, 242 (03) :C131-C145
[6]   EFFECT OF AMILORIDE AND SOME OF ITS ANALOGS ON CATION-TRANSPORT IN ISOLATED FROG SKIN AND THIN LIPID-MEMBRANES [J].
BENOS, DJ ;
SIMON, SA ;
MANDEL, LJ ;
CALA, PM .
JOURNAL OF GENERAL PHYSIOLOGY, 1976, 68 (01) :43-63
[7]  
BESTERMAN JM, 1985, J BIOL CHEM, V260, P1155
[8]   MEMBRANE ELECTRICAL-PROPERTIES OF VESICULAR NA-CA EXCHANGE INHIBITORS IN SINGLE ATRIAL MYOCYTES [J].
BIELEFELD, DR ;
HADLEY, RW ;
VASSILEV, PM ;
HUME, JR .
CIRCULATION RESEARCH, 1986, 59 (04) :381-389
[9]   EFFECTS OF SOME PYRAZINECARBOXAMIDES ON SODIUM-TRANSPORT IN FROG SKIN [J].
CUTHBERT, AW ;
FANELLI, GM .
BRITISH JOURNAL OF PHARMACOLOGY, 1978, 63 (01) :139-149
[10]   EVIDENCE FOR A NA+/H+ EXCHANGER AT THE BASOLATERAL MEMBRANES OF THE ISOLATED FROG-SKIN EPITHELIUM - EFFECT OF AMILORIDE ANALOGS [J].
EHRENFELD, J ;
CRAGOE, EJ ;
HARVEY, BJ .
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY, 1987, 409 (1-2) :200-207