SYNTHESIS AND ENZYMATIC EVALUATION OF PYRIDOSTIGMINE ANALOGS USED TO PROBE ACTIVE-SITES OF ACETYLCHOLINESTERASE AND BUTYRYLCHOLINESTERASE

被引：17

作者：

MILLNER, OE

STANLEY, JW

PURCELL, WP

机构：

[1] UNIV TENNESSEE,GRAD SCH MED SCI,MEMPHIS,TN 38163

[2] UNIV TENNESSEE,COLL PHARM,DEPT MOLEC & QUANTUM BIOL,MED UNITS,MEMPHIS,TN 38163

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1974年 / 17卷 / 01期

关键词：

D O I：

10.1021/jm00247a004

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：13 / 18

页数：6

共 25 条

[1] THE CHOLINESTERASES OF HUMAN BLOOD .2. THE FORCES ACTING BETWEEN ENZYME AND SUBSTRATE [J].

ADAMS, DH ;

WHITTAKER, VP .

BIOCHIMICA ET BIOPHYSICA ACTA, 1950, 4 (04) :543-558

[2] NATURE OF AN ANIONIC SITE IN BUTYRYLCHOLINESTERASE COMPARED WITH THAT OF A SIMILAR SITE IN ACETYLCHOLINESTERASE [J].

AUGUSTINSSON, KB .

BIOCHIMICA ET BIOPHYSICA ACTA, 1966, 128 (02) :351-+

[3]

AUGUSTINSSON KB, 1963, HDB EXPTL PHARMAKOLO, V15

[4] EFFECT OF PIPERIDINECARBOXAMIDE DERIVATIVES ON ISOLATED HUMAN PLASMA CHOLINESTERASE .2. VARIATIONS IN AMIDE FUNCTION [J].

BEASLEY, JG ;

QUINTANA, RP ;

NELMS, GG .

JOURNAL OF MEDICINAL CHEMISTRY, 1964, 7 (06) :698-&

[5]

BERGMANN F, 1958, ADV CATAL, V10, P131

[6] CHOLINESTERASE CATALYSIS [J].

BRESTKIN, AP ;

ROZENGAR.EV .

NATURE, 1965, 205 (4969) :388-&

[7]

CLAYTON JM, 1971, THESIS U TENNESSEE M

[8]

COHEN JA, 1963, HDB EXPTL PHARMAKOLO, V15

[9] CARBAMYLATION AND AFFINITY CONSTANTS OF SOME CARBAMATE INHIBITORS OFACETYLCHOLINESTERASE AND THEIR RELATION TO ANALOGOUS SUBSTRATE CONSTANTS [J].

HASTINGS, FL ;

MAIN, AR ;

IVERSON, F .

JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 1970, 18 (03) :497-+

[10]

KABACHNI.MI, 1970, PHARMACOL REV, V22, P355

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